SCHEMBL9178754

SCHEMBL9178754

Cc1cc(CCCOc2c(C)cc(C(=O)O)cc2C)on1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.57
NR1I2 O75469 1/20 0.57
CYP3A4 P08684 1/20 0.57
HCAR2 Q8TDS4 1/20 0.40
VHL P40337 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
PLA2G2A P14555 2/20 0.37
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
PPARA Q07869 1/20 0.35
BRD4 O60885 1/20 0.35
BRD2 P25440 1/20 0.35
CREBBP Q92793 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9201165 0.88 CYP2D6 (0.56) CYP2D6NR1I2CYP3A4HCAR2VHL
SCHEMBL8875268 0.88 CYP2D6 (0.56) CYP2D6NR1I2CYP3A4HCAR2VHL
SCHEMBL9863164 0.88 NR1I2 (0.46) CYP2D6NR1I2CYP3A4HCAR2VHL
SCHEMBL8875953 0.87 NR1I2 (0.55) CYP2D6NR1I2CYP3A4VHLMEN1
SCHEMBL10413141 0.87 PLAU (0.51) CYP2D6NR1I2CYP3A4HCAR2VHL
SCHEMBL9706268 0.87 NR1I2 (0.45) CYP2D6NR1I2CYP3A4HCAR2PLA2G2A
SCHEMBL9209739 0.86 NR1I2 (0.54) CYP2D6NR1I2CYP3A4VHLMEN1
SCHEMBL9202726 0.84 CYP2D6 (0.51) CYP2D6NR1I2CYP3A4HCAR2VHL
SCHEMBL9208970 0.83 NR1I2 (0.51) CYP2D6NR1I2CYP3A4VHLMEN1
SCHEMBL9862923 0.83 NR1I2 (0.45) CYP2D6NR1I2CYP3A4HCAR2VHL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5464848-A 1,2,4-oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC. (US) 1995-11-07 US disclosed
EP-0413289-B1 Oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC (US) 1995-02-01 EP disclosed
US-5110821-A Picornavirus STERLING DRUG INC. (US) 1992-05-05 US disclosed
EP-0413289-A2 Oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC. (US) 1991-02-20 EP disclosed