SCHEMBL9209739

SCHEMBL9209739

CCOC(=O)c1cc(C)c(OCCCc2cc(C)no2)c(C)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
RAB9A P51151 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
ESR1 P03372 2/20 0.40
BRD4 O60885 1/20 0.40
BRD2 P25440 1/20 0.40
CREBBP Q92793 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
LMNA P02545 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
ALDH1A1 P00352 3/20 0.38
THRB P10828 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8875953 0.89 NR1I2 (0.55) NR1I2CYP3A4CYP2D6RAB9AMEN1
SCHEMBL10413619 0.88 NR1I2 (0.44) NR1I2CYP3A4CYP2D6RAB9ATDP1
SCHEMBL9178754 0.86 CYP2D6 (0.57) NR1I2CYP3A4CYP2D6RAB9ABRD4
SCHEMBL9201165 0.85 CYP2D6 (0.56) NR1I2CYP3A4CYP2D6RAB9AMEN1
SCHEMBL8875268 0.85 CYP2D6 (0.56) NR1I2CYP3A4CYP2D6RAB9AMEN1
SCHEMBL8875936 0.85 NR1I2 (0.62) NR1I2CYP3A4CYP2D6RAB9ATDP1
SCHEMBL8874325 0.82 NR1I2 (0.48) NR1I2CYP3A4CYP2D6RAB9ATDP1
SCHEMBL9202726 0.81 CYP2D6 (0.51) NR1I2CYP3A4CYP2D6RAB9AMEN1
SCHEMBL5884654 0.80 NR1I2 (0.51) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL9208970 0.80 NR1I2 (0.51) NR1I2CYP3A4CYP2D6RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0413289-B1 Oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC (US) 1995-02-01 EP disclosed
US-5110821-A Picornavirus STERLING DRUG INC. (US) 1992-05-05 US disclosed
EP-0413289-A2 Oxadiazolyl-phenoxyalkylisoxazoles and their use as antiviral agents STERLING WINTHROP INC. (US) 1991-02-20 EP disclosed