SCHEMBL9181519

SCHEMBL9181519

C=C[C@H]1CC[C@H](C2CCC(c3ccc(Cl)c(Cl)c3)CC2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 11/20 0.43
SLC6A4 P31645 11/20 0.43
SLC6A3 Q01959 11/20 0.43
KCNH2 Q12809 8/20 0.43
CYP2D6 P10635 8/20 0.43
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
MLNR O43193 1/20 0.35
NR1I2 O75469 1/20 0.35
ABCB11 O95342 1/20 0.35
ESR1 P03372 1/20 0.35
CYP1A2 P05177 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
ABCB1 P08183 1/20 0.35
ADRB1 P08588 1/20 0.35
CYP3A4 P08684 1/20 0.35
HTR1A P08908 1/20 0.35
CHRM5 P08912 1/20 0.35
ADRA2A P08913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9181525 1.00 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL9628787 1.00 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL9181582 0.86 SLC6A2 (0.33) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL14274436 0.86 SLC6A2 (0.33) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL9181594 0.86 SLC6A2 (0.33) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL9181599 0.86 SLC6A2 (0.33) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL11046032 0.83 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL11046036 0.83 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL8380296 0.83 AHR (0.44) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6
SCHEMBL8380293 0.83 AHR (0.44) SLC6A2SLC6A4SLC6A3KCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458176-B1 Bicyclohexyl derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 EP disclosed
US-5174921-A BICYCLOHEXYL DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 1992-12-29 US disclosed
EP-0458176-A1 Bicyclohexyl derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-11-27 EP disclosed