SCHEMBL9181582

SCHEMBL9181582

C=C[C@H]1CC[C@H](C2CCC(c3ccc(Cl)c(F)c3)CC2)CC1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 5/20 0.33
SLC6A4 P31645 5/20 0.33
SLC6A3 Q01959 5/20 0.33
CYP2D6 P10635 2/20 0.31
KCNH2 Q12809 2/20 0.31
RIPK1 Q13546 1/20 0.31
HSD11B1 P28845 1/20 0.30
HTR7 P34969 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9181594 1.00 SLC6A2 (0.33) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL14274436 1.00 SLC6A2 (0.33) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL9181599 1.00 SLC6A2 (0.33) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2
SCHEMBL9135342 0.92 OPRL1 (0.34) SLC6A2SLC6A4SLC6A3
SCHEMBL8518707 0.87 OPRL1 (0.36) SLC6A2SLC6A4SLC6A3HSD11B1
SCHEMBL6461351 0.87 SLC6A2 (0.32) SLC6A2SLC6A4SLC6A3
SCHEMBL8518711 0.87 OPRL1 (0.36) SLC6A2SLC6A4SLC6A3HSD11B1
SCHEMBL8518709 0.87 OPRL1 (0.36) SLC6A2SLC6A4SLC6A3HSD11B1
SCHEMBL6461349 0.87 SLC6A2 (0.32) SLC6A2SLC6A4SLC6A3
SCHEMBL9628787 0.86 SLC6A2 (0.43) SLC6A2SLC6A4SLC6A3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458176-B1 Bicyclohexyl derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 EP claimed
EP-0458176-B1 Bicyclohexyl derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 EP disclosed
US-5174921-A BICYCLOHEXYL DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 1992-12-29 US disclosed
EP-0458176-A1 Bicyclohexyl derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-11-27 EP disclosed