SCHEMBL9187166

SCHEMBL9187166

CCCC(F)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.44
SLC6A4 P31645 2/20 0.41
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
MC4R P32245 1/20 0.38
CYP19A1 P11511 1/20 0.37
CYP3A4 P08684 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
ACP3 P15309 1/20 0.36
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
FFAR1 O14842 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27528113 0.83 PDE2A (0.47) PDE2ACES2CES1MC4RCA1
SCHEMBL16976289 0.82 PDE2A (0.46) PDE2ASLC6A4CES2CES1MC4R
SCHEMBL2090318 0.80 PDE2A (0.49) PDE2ASLC6A4CES2CES1MC4R
SCHEMBL2763340 0.78 HSD11B1 (0.47) PDE2ASLC6A4CES2CES1CYP3A4
SCHEMBL906186 0.78 HSD11B1 (0.47) PDE2ASLC6A4CES2CES1CYP3A4
SCHEMBL3612320 0.78 PDE2A (0.43) PDE2ASLC6A4CES2CES1MC4R
SCHEMBL3602797 0.78 PDE2A (0.43) PDE2ASLC6A4MC4R
SCHEMBL2764096 0.78 PDE2A (0.43) PDE2ASLC6A4CES2CES1MC4R
SCHEMBL16230332 0.78 PDE2A (0.43) PDE2ASLC6A4CES2CES1MC4R
SCHEMBL3595268 0.78 PDE2A (0.43) PDE2ASLC6A4MC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674651-A1 SUBSTITUTED 6-AZAANDROSTENONES GLAXO WELLCOME INC. (US) 1995-10-04 EP disclosed