SCHEMBL9190836

SCHEMBL9190836

CC(C)C(c1ccc2nccnc2c1)n1ccnc1

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 7/20 0.57
CYP11B1 P15538 3/20 0.53
CYP11B2 P19099 3/20 0.53
CYP19A1 P11511 2/20 0.44
OGA O60502 5/20 0.43
CYP26A1 O43174 4/20 0.42
CYP3A4 P08684 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9192264 0.78 CYP17A1 (0.49) CYP17A1CYP11B1CYP11B2CYP19A1CYP26A1
SCHEMBL9078342 0.78 CYP17A1 (0.58) CYP17A1CYP11B1CYP11B2CYP19A1CYP26A1
SCHEMBL7457164 0.76 CYP17A1 (0.50) CYP17A1CYP11B1CYP11B2CYP19A1CYP26A1
SCHEMBL9198992 0.76 CYP11B1 (0.47) CYP17A1CYP11B1CYP11B2CYP19A1CYP26A1
SCHEMBL9198062 0.76 CYP11B1 (0.47) CYP17A1CYP11B1CYP11B2CYP19A1CYP26A1
SCHEMBL9196154 0.75 CYP19A1 (0.69) CYP17A1CYP11B1CYP11B2CYP19A1CYP26A1
SCHEMBL4054853 0.75 CYP17A1 (0.68) CYP17A1CYP11B1CYP11B2CYP19A1CYP26A1
SCHEMBL9199149 0.74 CYP19A1 (0.72) CYP17A1CYP11B1CYP11B2CYP19A1CYP26A1
Oxalic Acid SCHEMBL9663654 0.74 CYP17A1 (0.48) CYP17A1CYP11B1CYP11B2CYP19A1CYP26A1
Hydrochloric Acid SCHEMBL9079014 0.74 CYP17A1 (0.48) CYP17A1CYP11B1CYP11B2CYP19A1CYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1036003-C A process for preparing (1H-azol-1-ylmethyl) substituted quinoxaline derivatives JANSSEN PHARMACEUTICA NV (BE) 1997-10-01 CN disclosed
CN-1033752-C (1H-azol-1-ylmethyl) substituted quinoline or quinolinone derivatives JANSSEN PHARMACEUTICA NV (SE) 1997-01-08 CN disclosed
EP-0371564-B1 (1H-azol-1-ylmethyl)substituted quinoline, quinazoline or quinoxaline derivatives JANSSEN PHARMACEUTICA NV (BE) 1995-07-12 EP disclosed
US-5151421-A Compounds for inhibition of metabolism of retinoids, for treatment for proliferation of epithelial cells and keratin disorders JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-29 US disclosed
US-5028606-A Retinoid metabolism inhibitors JANSSEN PHARMACEUTICA N.V. (BE) 1991-07-02 US disclosed