SCHEMBL9192054

SCHEMBL9192054

CCC(=O)c1cnc(Cl)c(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.46
ALDH1A1 P00352 7/20 0.45
MAPK1 P28482 2/20 0.45
TDP1 Q9NUW8 4/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
NPSR1 Q6W5P4 2/20 0.42
MEN1 O00255 3/20 0.42
RXFP1 Q9HBX9 1/20 0.42
KDM4E B2RXH2 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9198640 0.84 PPARA (0.38) KMT2AALDH1A1MAPK1TDP1L3MBTL1
SCHEMBL6133961 0.83 GSK3B (0.48) KMT2AALDH1A1MAPK1TDP1L3MBTL1
SCHEMBL15003979 0.83 HSD17B3 (0.45) KMT2AALDH1A1MAPK1TDP1L3MBTL1
SCHEMBL9197903 0.82 ALDH1A1 (0.43) KMT2AALDH1A1
SCHEMBL9193384 0.82 CYP2D6 (0.45) ALDH1A1KDM4E
SCHEMBL9841175 0.81 ALDH1A1 (0.43) KMT2AALDH1A1MAPK1TDP1L3MBTL1
SCHEMBL4285053 0.81 GSK3B (0.50) KMT2AALDH1A1MAPK1TDP1L3MBTL1
Hydrochloric Acid SCHEMBL9722613 0.80 ALDH1A1 (0.43) KMT2AALDH1A1MAPK1TDP1L3MBTL1
SCHEMBL27931887 0.80 MEN1 (0.49) KMT2AALDH1A1MAPK1TDP1L3MBTL1
SCHEMBL27913968 0.80 HTT (0.44) KMT2AALDH1A1MAPK1MEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3356387-B1 ANTIMICROBIAL POLYMYXIN DERIVATIVE COMPOUNDS UNIV MONASH (AU) 2024-06-26 EP disclosed
CN-101932570-B TRPV1 antagonists and uses thereof PURDUE PHARMA LP 2014-11-26 CN disclosed
CN-101932570-A The TRPV1 antagonist with and uses thereof SHIONOGI & CO 2010-12-29 CN disclosed
EP-0299277-B1 Process for the preparation of substituted pyridyl-alkyl ketones BAYER AG (DE) 1995-10-18 EP disclosed
US-4990620-A Halogen substituted pyridylalkyl ketones BAYER AKTIENGESELLSCHAFT (DE) 1991-02-05 US disclosed
US-4927938-A Halogen substituted pyridylalkyl ketones BAYER AKTIENGESELLSCHAFT (DE) 1990-05-22 US disclosed
EP-0299277-A2 Process for the preparation of substituted pyridyl-alkyl ketones BAYER AG (DE) 1989-01-18 EP disclosed