SCHEMBL9193003

SCHEMBL9193003

COC(=O)C(=CN(C)C)N(C)c1cccc(Br)n1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 1/20 0.38
GRM5 P41594 1/20 0.32
HTR7 P34969 1/20 0.32
NCEH1 Q6PIU2 2/20 0.31
PKM P14618 1/20 0.31
HTR1A P08908 1/20 0.31
FGFR4 P22455 2/20 0.31
CHRNB2 P17787 2/20 0.30
CHRNA4 P43681 2/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9158190 0.89 CLK1 (0.39) CLK1GRM5HTR7NCEH1PKM
SCHEMBL9865275 0.86 CLK1 (0.38) CLK1GRM5HTR7NCEH1PKM
SCHEMBL9158184 0.86 CLK1 (0.38) CLK1GRM5HTR7NCEH1PKM
SCHEMBL8734918 0.86 CLK1 (0.38) CLK1GRM5HTR7NCEH1PKM
SCHEMBL9191662 0.78 CNR1 (0.45)
SCHEMBL9550193 0.78 CNR1 (0.45)
SCHEMBL9030991 0.74 ALDH1A1 (0.38) ALDH1A1HPGD
SCHEMBL9469921 0.74 ALDH1A1 (0.38) ALDH1A1HPGD
SCHEMBL17804225 0.73 CLK1 (0.40) CLK1GRM5HTR7NCEH1PKM
SCHEMBL1400663 0.73 CLK1 (0.40) CLK1GRM5HTR7NCEH1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0471262-B1 Process for the production of substituted 3-amino-acrylesters BAYER AG (DE) 1995-11-15 EP disclosed
US-5196541-A PROCESS FOR THE PREPARATION OF SUBSTITUTED 3-AMINOACRYLIC ESTERS BAYER AKTIENGESELLSCHAFT (DE) 1993-03-23 US disclosed
EP-0471262-A1 Process for the production of substituted 3-amino-acrylesters BAYER AG (DE) 1992-02-19 EP disclosed