SCHEMBL9194271

SCHEMBL9194271

O=C1CC2(C(=O)N1)c1ccccc1CCc1ccccc12

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.44
MAPK13 O15264 1/20 0.44
MAPK12 P53778 1/20 0.44
MAPK11 Q15759 1/20 0.44
MAPK14 Q16539 1/20 0.44
TSHR P16473 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
AKR1B1 P15121 1/20 0.41
HTR2A P28223 1/20 0.40
MAPT P10636 1/20 0.38
SRD5A1 P18405 1/20 0.38
AHR P35869 1/20 0.37
PDK2 Q15119 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9673557 0.81 AKR1B1 (0.45) AKR1B1
SCHEMBL10970579 0.76 ALOX5 (0.36) AKR1B1
SCHEMBL10834099 0.76 PDK2 (0.50) TDP1AKR1B1MAPTPDK2
SCHEMBL7416528 0.75 TSHR (0.49) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL5107203 0.73 GSK3B (0.43) AKR1B1
SCHEMBL10971658 0.73 AKR1B1 (0.51) TSHRTDP1AKR1B1HTR2AMAPT
SCHEMBL10970570 0.72 BACE1 (0.43) TSHRTDP1AKR1B1HTR2AMAPT
SCHEMBL30364417 0.71 TSHR (0.49) NPC1MAPK13MAPK12MAPK11MAPK14
SCHEMBL9672258 0.70 PDK2 (0.44) TDP1PDK2
SCHEMBL22904131 0.70 CYP19A1 (0.36) AKR1B1PDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456183-B1 Spiro dibenzosuberane derivatives SHIONOGI & CO (JP) 1995-10-04 EP disclosed
EP-0456183-A2 Spiro dibenzosuberane derivatives SHIONOGI SEIYAKU KABUSHIKI KAISHA (JP) 1991-11-13 EP disclosed