SCHEMBL9196121

SCHEMBL9196121

COc1ccc(CCSC(=N)N)cc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 5/20 0.72
CYP2D6 P10635 3/20 0.72
NPC1 O15118 1/20 0.72
CYP3A4 P08684 1/20 0.72
RAB9A P51151 1/20 0.72
HIF1A Q16665 1/20 0.72
IDO1 P14902 4/20 0.72
BLM P54132 1/20 0.70
NPSR1 Q6W5P4 1/20 0.70
TAAR1 Q96RJ0 1/20 0.56
NOS3 P29474 1/20 0.56
NOS2 P35228 1/20 0.56
LMNA P02545 1/20 0.54
ALDH1A1 P00352 2/20 0.53
CYP1A2 P05177 2/20 0.53
MEN1 O00255 1/20 0.53
TP53 P04637 1/20 0.53
MAPT P10636 1/20 0.53
ALOX15 P16050 1/20 0.53
MAPK1 P28482 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4316762 0.85 NOS1 (1.00) NOS1CYP2D6NPC1CYP3A4RAB9A
SCHEMBL5045935 0.84 IDO1 (1.00) NOS1CYP2D6IDO1NOS3NOS2
SCHEMBL9193560 0.83 NOS1 (0.68) NOS1CYP2D6NPC1CYP3A4RAB9A
Bromide SCHEMBL2283156 0.83 BLM (1.00) NOS1CYP2D6NPC1CYP3A4RAB9A
Hydrochloric Acid SCHEMBL489767 0.82 IDO1 (1.00) NOS1CYP2D6IDO1NOS3NOS2
SCHEMBL8061071 0.82 NOS1 (0.70) NOS1CYP2D6NPC1CYP3A4RAB9A
SCHEMBL26313245 0.80 NOS1 (0.81) NOS1CYP2D6NPC1CYP3A4RAB9A
SCHEMBL26313250 0.80 NOS1 (0.81) NOS1CYP2D6NPC1CYP3A4RAB9A
SCHEMBL26313697 0.80 NOS1 (0.81) NOS1CYP2D6NPC1CYP3A4RAB9A
SCHEMBL13067607 0.80 NOS1 (0.88) NOS1CYP2D6NPC1CYP3A4RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0670720-A1 ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-09-13 EP claimed
WO-1994012165-A2 ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1994-06-09 WO claimed
EP-0670720-A1 ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1995-09-13 EP disclosed
WO-1994012165-A2 ENZYME INHIBITORS THE WELLCOME FOUNDATION LIMITED (GB) 1994-06-09 WO disclosed