SCHEMBL9196331

SCHEMBL9196331

N#Cc1ccc(C(CCc2ccc(F)cc2)n2cnnn2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 15/20 0.68
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
SLC1A2 P43004 1/20 0.38
KCNH2 Q12809 1/20 0.38
CACNA1F O60840 1/20 0.38
HTR1A P08908 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
DRD2 P14416 1/20 0.38
DRD1 P21728 1/20 0.38
DRD4 P21917 1/20 0.38
DRD5 P21918 1/20 0.38
HRH2 P25021 1/20 0.38
ADRA1D P25100 1/20 0.38
HTR2A P28223 1/20 0.38
HTR7 P34969 1/20 0.38
ADRA1A P35348 1/20 0.38
HRH1 P35367 1/20 0.38
ADRA1B P35368 1/20 0.38
OPRM1 P35372 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104838 0.81 CYP19A1 (1.00) CYP19A1CYP11B1CYP11B2
SCHEMBL9191150 0.79 CYP19A1 (0.65) CYP19A1SLC1A2KCNH2CACNA1FHTR1A
SCHEMBL8408606 0.76 CYP19A1 (1.00) CYP19A1
SCHEMBL8102936 0.74 CYP19A1 (1.00) CYP19A1CYP11B1CYP11B2
SCHEMBL2348017 0.72 CYP19A1 (0.61) CYP19A1CYP11B1CYP11B2
SCHEMBL9194497 0.71 CYP19A1 (0.54) CYP19A1CYP11B1CYP11B2SLC1A2KCNH2
SCHEMBL8104816 0.71 CYP19A1 (0.54) CYP19A1CYP11B1CYP11B2SLC1A2KCNH2
SCHEMBL8109000 0.71 CYP19A1 (0.54) CYP19A1SLC1A2KCNH2CACNA1FHTR1A
SCHEMBL8110779 0.70 CYP19A1 (1.00) CYP19A1CYP11B1CYP11B2
SCHEMBL8104979 0.68 CYP19A1 (0.72) CYP19A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0674626-A1 NOVEL SELECTIVE AROMATASE INHIBITING COMPOUNDS ORION-YHTYMÄ OY (FI) 1995-10-04 EP claimed
WO-1994013645-A1 NOVEL SELECTIVE AROMATASE INHIBITING COMPOUNDS Orion-Yhtymä Oy (FI) 1994-06-23 WO claimed
EP-0674626-A1 NOVEL SELECTIVE AROMATASE INHIBITING COMPOUNDS ORION-YHTYMÄ OY (FI) 1995-10-04 EP disclosed
WO-1994013645-A1 NOVEL SELECTIVE AROMATASE INHIBITING COMPOUNDS Orion-Yhtymä Oy (FI) 1994-06-23 WO disclosed