SCHEMBL9201604

SCHEMBL9201604

CCN(CCO)CCNc1cc(=O)n(C)c(=O)n1C

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.60
ADRB1 P08588 2/20 0.59
SLC6A4 P31645 2/20 0.59
SLC22A2 O15244 1/20 0.59
KCNH2 Q12809 1/20 0.59
SLC47A2 Q86VL8 1/20 0.59
SLC47A1 Q96FL8 1/20 0.59
CYP1A2 P05177 1/20 0.57
NPSR1 Q6W5P4 2/20 0.52
HSD17B10 Q99714 2/20 0.52
TSHR P16473 2/20 0.52
POLB P06746 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
TAAR1 Q96RJ0 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.45
HPGD P15428 1/20 0.45
ALDH1A1 P00352 3/20 0.44
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9205218 0.81 MAPK1 (0.72) MAPK1ADRB1SLC6A4SLC22A2KCNH2
SCHEMBL9429589 0.80 ADRB1 (0.75) MAPK1ADRB1SLC6A4SLC22A2KCNH2
SCHEMBL8780899 0.79 TAAR1 (0.67) MAPK1ADRB1SLC6A4SLC22A2KCNH2
SCHEMBL9428809 0.79 ADRB1 (0.71) MAPK1ADRB1SLC6A4SLC22A2KCNH2
SCHEMBL9429159 0.79 TAAR1 (0.48) MAPK1ADRB1SLC6A4SLC22A2KCNH2
SCHEMBL9428920 0.78 SLC22A2 (0.56) MAPK1ADRB1SLC6A4SLC22A2KCNH2
Oxalic Acid SCHEMBL9428776 0.78 TAAR1 (0.62) MAPK1ADRB1SLC6A4SLC22A2KCNH2
SCHEMBL9428818 0.78 ADRB1 (0.64) MAPK1ADRB1SLC6A4SLC22A2KCNH2
SCHEMBL9429051 0.78 CYP1A2 (0.51) MAPK1ADRB1SLC6A4SLC22A2KCNH2
SCHEMBL9428374 0.78 ADRB1 (0.75) MAPK1ADRB1SLC6A4SLC22A2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0430693-B1 Pyrimidinedione derivative compounds, method for preparing same, and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS (JP) 1995-05-31 EP disclosed
US-5114941-A PYRIMIDINEDIONE DERIVATIVE COMPOUNDS, METHOD FOR PREPARING SAME, AND ANTIARRYTHMIC AGENTS CONTAINING SAME MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1992-05-19 US disclosed
EP-0430693-A2 Pyrimidinedione derivative compounds, method for preparing same, and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-06-05 EP disclosed