SCHEMBL9201626

SCHEMBL9201626

CS(=O)(=O)c1ccc(-c2cc(C(=O)N3CCCC3)nn2-c2ccc(F)cc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.67
CHRNA7 P36544 2/20 0.65
MALT1 Q9UDY8 1/20 0.64
AOC3 Q16853 1/20 0.60
PTGS1 P23219 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9208534 0.92 PTGS2 (0.65) PTGS2CHRNA7MALT1AOC3PTGS1
SCHEMBL9210924 0.84 AOC3 (0.70) PTGS2CHRNA7AOC3PTGS1
SCHEMBL9203245 0.84 MEN1 (0.70) PTGS2CHRNA7AOC3PTGS1
SCHEMBL27524813 0.84 AOC3 (0.61) PTGS2CHRNA7AOC3PTGS1
SCHEMBL9201596 0.84 MALT1 (0.65) PTGS2CHRNA7MALT1
SCHEMBL16640301 0.83 MALT1 (0.67) PTGS2CHRNA7MALT1PTGS1
SCHEMBL9199556 0.83 AOC3 (0.65) PTGS2CHRNA7AOC3PTGS1
SCHEMBL9204761 0.83 AOC3 (0.65) PTGS2CHRNA7AOC3PTGS1
SCHEMBL9055103 0.82 AOC3 (0.64) PTGS2CHRNA7AOC3PTGS1
SCHEMBL16640303 0.82 MALT1 (0.65) PTGS2CHRNA7MALT1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1046506-C Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1999-11-17 CN disclosed
EP-0418845-B1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1995-08-09 EP disclosed
US-5134142-A PYRAZOLE DERIVATIVES, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-07-28 US disclosed
EP-0418845-A1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-03-27 EP disclosed