SCHEMBL9201792

SCHEMBL9201792

CSc1ccc(-n2nc(C#N)cc2-c2ccc(F)cc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.63
NR3C2 P08235 1/20 0.51
PTGS1 P23219 5/20 0.46
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ATM Q13315 1/20 0.41
KDM1A O60341 1/20 0.39
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
AOC3 Q16853 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9209095 1.00 PTGS2 (0.63) PTGS2NR3C2PTGS1MEN1KMT2A
Hydrochloric Acid SCHEMBL9199123 0.85 PTGS2 (0.46) PTGS2NR3C2PTGS1MEN1KMT2A
Hydrochloric Acid SCHEMBL9207583 0.84 PTGS2 (0.46) PTGS2NR3C2PTGS1MEN1KMT2A
SCHEMBL9207196 0.84 PTGS2 (0.46) PTGS2NR3C2PTGS1MEN1KMT2A
SCHEMBL9202425 0.84 PTGS2 (0.48) PTGS2NR3C2PTGS1KDM1A
SCHEMBL9210967 0.84 PTGS2 (0.69) PTGS2NR3C2PTGS1MEN1KMT2A
SCHEMBL9207646 0.83 PTGS2 (0.65) PTGS2NR3C2PTGS1
SCHEMBL8641979 0.83 PTGS2 (0.45) PTGS2NR3C2PTGS1
SCHEMBL8642066 0.83 PTGS2 (0.47) PTGS2NR3C2PTGS1
SCHEMBL9207835 0.82 PTGS2 (0.51) PTGS2PTGS1MEN1KMT2AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0418845-B1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1995-08-09 EP disclosed
US-5134142-A PYRAZOLE DERIVATIVES, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-07-28 US disclosed
EP-0418845-A1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-03-27 EP disclosed