SCHEMBL9201844

SCHEMBL9201844

CCc1nc2ncc(C)c(C)c2[nH]1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 5/20 0.53
ADORA3 P0DMS8 4/20 0.43
ADORA2A P29274 3/20 0.43
PI4KA P42356 1/20 0.36
PI4K2B Q8TCG2 1/20 0.36
PI4K2A Q9BTU6 1/20 0.36
PI4KB Q9UBF8 1/20 0.36
DDAH1 O94760 1/20 0.33
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
GAA P10253 1/20 0.32
HTT P42858 1/20 0.32
TP53 P04637 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3211252 0.75 ADORA1 (0.57) ADORA1ADORA3ADORA2API4KAPI4K2B
SCHEMBL9137080 0.74 ADORA1 (0.38) ADORA1ADORA3ADORA2ACCNA2CDK2
SCHEMBL21305258 0.73 ADORA1 (0.50) ADORA1ADORA3ADORA2API4KAPI4K2B
SCHEMBL9406903 0.70 PI4KA (0.44) ADORA1ADORA3ADORA2API4KAPI4K2B
SCHEMBL5091129 0.69 ADORA1 (1.00) ADORA1ADORA3ADORA2ADDAH1NOS3
SCHEMBL9847095 0.69 ADORA1 (0.46) ADORA1ADORA3ADORA2ADDAH1GAA
SCHEMBL23178669 0.69 ADORA1 (0.40) ADORA1ADORA3ADORA2API4KAPI4K2B
SCHEMBL9406713 0.68 ADORA1 (0.41) ADORA1ADORA3ADORA2API4KAPI4K2B
SCHEMBL9406510 0.68 PI4KA (0.52) ADORA3ADORA2API4KAPI4K2BPI4K2A
SCHEMBL31569181 0.68 KDM4E (0.41) ADORA1PI4KAPI4K2BPI4K2API4KB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0517812-A4 ANGIOTENSIN II ANTAGONISTS INCORPORATING A SUBSTITUTED BENZYL ELEMENT MERCK & CO INC (US) 1995-10-18 EP disclosed
EP-0517812-A1 ANGIOTENSIN II ANTAGONISTS INCORPORATING A SUBSTITUTED BENZYL ELEMENT MERCK & CO. INC. (US) 1992-12-16 EP disclosed
EP-0456510-A1 Antihypertensive products, a process for their preparation and pharamaceutical compositions containing them MERCK & CO. INC. (US) 1991-11-13 EP disclosed