SCHEMBL9205089

SCHEMBL9205089

CC[C@@](C)(C(=O)O)[C@](C)(Br)C(=O)O

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.35
ALDH1A1 P00352 2/20 0.35
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
HIF1A Q16665 1/20 0.33
GRM2 Q14416 1/20 0.31
GRM3 Q14832 1/20 0.31
MEN1 O00255 2/20 0.31
CYP1A2 P05177 2/20 0.31
KMT2A Q03164 2/20 0.31
THRB P10828 1/20 0.31
FFAR3 O14843 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9212741 0.81 ALDH1A1 (0.32) TSHRALDH1A1CYP2D6CYP2C19HIF1A
SCHEMBL9154668 0.81 TSHR (0.44) TSHRALDH1A1CYP2D6CYP2C19HIF1A
SCHEMBL9203463 0.78 AKR1B1 (0.33) TSHRALDH1A1MEN1KMT2A
SCHEMBL284018 0.76 TSHR (0.40) TSHRALDH1A1CYP2D6CYP2C19HIF1A
Ammonia Solution, Strong SCHEMBL28651755 0.74 TSHR (0.38) TSHRALDH1A1CYP2D6CYP2C19HIF1A
SCHEMBL10830599 0.74 TSHR (0.38) TSHRALDH1A1CYP2D6CYP2C19HIF1A
SCHEMBL9710097 0.74 TSHR (0.38) TSHRALDH1A1CYP2D6CYP2C19HIF1A
SCHEMBL28727403 0.74 TSHR (0.38) TSHRALDH1A1CYP2D6CYP2C19HIF1A
SCHEMBL5274369 0.72 TSHR (0.36) TSHRALDH1A1CYP2D6CYP2C19HIF1A
SCHEMBL800011 0.72 ALDH1A1 (0.36) TSHRALDH1A1CYP2D6CYP2C19HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0643710-A1 SYNTHESIS OF OPTICALLY ACTIVE LACTONES FROM L-ASPARTIC ACID AND INTERMEDIATES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-03-22 EP disclosed
US-5322942-A Deprotecting and hydrolyzing protected aspartic acid diester, reacting with nitrosylating agent in presence of hydrogen halide, esterifying, reacting with acyl aryl derivative REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1994-06-21 US disclosed
WO-1992021675-A1 SYNTHESIS OF OPTICALLY ACTIVE LACTONES FROM L-ASPARTIC ACID AND INTERMEDIATES THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1992-12-10 WO disclosed