SCHEMBL9205143

SCHEMBL9205143

CCCCc1nc(N)[nH]c(=O)c1Cc1ccc(-c2ccccc2)c(C#N)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.39
XDH P47989 1/20 0.39
CCR2 P41597 4/20 0.39
CCR5 P51681 1/20 0.39
HIF1A Q16665 1/20 0.38
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GALR3 O60755 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
ACHE P22303 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27771400 0.90 KDM4E (0.41) CYP19A1XDHPDE3BPDE3AKDM4E
SCHEMBL8671011 0.89 ACHE (0.45) HIF1AACHE
SCHEMBL28781819 0.89 CYP19A1 (0.39) CYP19A1XDHPDE3BPDE3AKDM4E
SCHEMBL27845844 0.88 CYP19A1 (0.40) CYP19A1CCR2CCR5PDE3BPDE3A
SCHEMBL27771428 0.88 CYP19A1 (0.39) CYP19A1PDE3BPDE3AKDM4EGALR3
SCHEMBL27845843 0.87 PPARG (0.43) CYP19A1PDE3BPDE3AKDM4EGALR3
SCHEMBL27771475 0.87 CYP19A1 (0.38) CYP19A1PDE3BPDE3AKDM4EGALR3
SCHEMBL27771413 0.87 BRS3 (0.39) CYP19A1PDE3BPDE3AKDM4EGALR3
SCHEMBL27771371 0.85 ACHE (0.38) CYP19A1CCR2CCR5PDE3BPDE3A
SCHEMBL27771424 0.85 CYP19A1 (0.37) CYP19A1PDE3BPDE3AKDM4EGALR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0680480-A1 PYRIMIDINONE DERIVATIVES FUSED TO NITROGEN HETEROCYCLES HAVING A II ANTAGONISTIC ACTIVITY. LUSO FARMACO INST (IT) 1995-11-08 EP disclosed