SCHEMBL9205342

SCHEMBL9205342

Cc1cc2c(cc1C)CC(=O)N(CCC1CCCCN1CCCc1ccncc1)CC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
HRH3 Q9Y5N1 4/20 0.37
HCN4 Q9Y3Q4 2/20 0.36
MAPT P10636 1/20 0.36
CYP3A4 P08684 2/20 0.35
ALOX15 P16050 1/20 0.35
ACHE P22303 1/20 0.34
GFER P55789 1/20 0.33
CHRNB1 P11230 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNB3 Q05901 1/20 0.33
CYP19A1 P11511 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
ALDH1A1 P00352 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9206942 0.88 KDM4E (0.35) KDM4EHRH3HCN4MAPTCYP3A4
Hydrochloric Acid SCHEMBL9740720 0.87 KDM4E (0.34) KDM4EHRH3HCN4MAPTCYP3A4
Hydrochloric Acid SCHEMBL9739345 0.85 HRH3 (0.40) HRH3CYP3A4CHRNB1CHRNB2CHRNB4
SCHEMBL9215931 0.84 HRH3 (0.38) KDM4EHRH3CYP3A4ACHECHRNB1
SCHEMBL9212354 0.82 HRH3 (0.35) KDM4EHRH3ACHEGFERCHRNB1
Hydrochloric Acid SCHEMBL9741088 0.81 HRH3 (0.34) KDM4EHRH3ACHEGFERCHRNB1
SCHEMBL9208353 0.81 HRH3 (0.42) HRH3CYP3A4CHRNB1CHRNB2CHRNB4
SCHEMBL9217265 0.79 DRD4 (0.43) HRH3HTR1ADRD3
SCHEMBL9214421 0.78 HRH3 (0.40) HRH3KCNH2
Hydrochloric Acid SCHEMBL9208307 0.76 HRH3 (0.39) HRH3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed