SCHEMBL9206728

SCHEMBL9206728

O/C1=C/c2ccccc2/C=C\c2ccc(Br)cc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRC P08575 2/20 0.35
BCL2 P10415 1/20 0.34
MCL1 Q07820 1/20 0.34
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
ALOX15 P16050 2/20 0.32
CYP2A6 P11509 1/20 0.32
MAPK1 P28482 2/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
GLA P06280 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
GPR84 Q9NQS5 1/20 0.32
GSTA1 P08263 1/20 0.32
S100A4 P26447 1/20 0.31
P2RX4 Q99571 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9206731 1.00 PTPRC (0.35) PTPRCBCL2MCL1ESR1ESR2
SCHEMBL9205323 0.88 PTPRC (0.34) PTPRCBCL2MCL1ALOX15CYP2A6
SCHEMBL9207295 0.88 PTPRC (0.34) PTPRCBCL2MCL1ALOX15CYP2A6
SCHEMBL9205329 0.88 PTPRC (0.34) PTPRCBCL2MCL1ALOX15CYP2A6
SCHEMBL9207293 0.88 PTPRC (0.34) PTPRCBCL2MCL1ALOX15CYP2A6
SCHEMBL9203655 0.86 PTPRC (0.35) PTPRCBCL2MCL1ESR1ESR2
SCHEMBL9203647 0.86 PTPRC (0.35) PTPRCBCL2MCL1ESR1ESR2
SCHEMBL9207972 0.78 GPR84 (0.42) PTPRCALOX15MAPK1KDM4ELMNA
SCHEMBL9207977 0.78 GPR84 (0.42) PTPRCALOX15MAPK1KDM4ELMNA
SCHEMBL9212754 0.72 PTPRC (0.42) PTPRCALOX15CYP2A6MAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0319073-B1 Cyclo-octane neuroprotective agents MERCK SHARP & DOHME (GB) 1995-08-23 EP disclosed
US-4927819-A ANTICONVULSANT, PREVENTION OF NEURODEGENERATIVE DISORDERS MERCK SHARP & DOHME LIMITED (GB) 1990-05-22 US disclosed
EP-0319073-A2 Cyclo-octane neuroprotective agents MERCK SHARP & DOHME LTD. (GB) 1989-06-07 EP disclosed