SCHEMBL9207296

SCHEMBL9207296

COc1ccc(-c2cc(C#N)nn2-c2ccc(OC)cc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.59
PTGS1 P23219 4/20 0.59
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C9 P11712 1/20 0.53
TSHR P16473 1/20 0.53
CYP2C19 P33261 1/20 0.53
THPO P40225 1/20 0.53
BLM P54132 1/20 0.53
PMP22 Q01453 1/20 0.53
HIF1A Q16665 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
RPA1 P27694 1/20 0.52
ALOX5 P09917 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9207646 0.93 PTGS2 (0.65) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL9208260 0.93 PTGS2 (0.64) PTGS2PTGS1CYP1A2CYP3A4CYP2C9
SCHEMBL5171748 0.90 PTGS2 (0.50) PTGS2PTGS1
Hydrochloric Acid SCHEMBL5147858 0.89 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL14504415 0.89 PTGS1 (0.49) PTGS2PTGS1RPA1ALOX5
SCHEMBL9210069 0.89 PTGS2 (0.60) PTGS2PTGS1ALOX5
SCHEMBL6340846 0.88 PTGS2 (0.75) PTGS2PTGS1
SCHEMBL9207837 0.88 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL14504421 0.88 PTGS1 (0.48) PTGS2PTGS1ALOX5
SCHEMBL9210134 0.88 PTGS2 (0.48) PTGS2PTGS1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0418845-B1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO (JP) 1995-08-09 EP disclosed
US-5134142-A PYRAZOLE DERIVATIVES, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1992-07-28 US disclosed
EP-0418845-A1 Pyrazole derivatives, processes for preparation thereof and pharmaceutical composition comprising the same FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-03-27 EP disclosed