SCHEMBL9209062

SCHEMBL9209062

O=c1c2ccccc2ccc2c(Cl)cccc12

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.61
CYP1A2 P05177 4/20 0.61
PAX8 Q06710 1/20 0.47
HPRT1 P00492 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
AKR1B1 P15121 2/20 0.44
CYP1A1 P04798 2/20 0.43
CYP1B1 Q16678 2/20 0.43
TDP1 Q9NUW8 2/20 0.42
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NR4A2 P43354 1/20 0.42
TP53 P04637 1/20 0.42
TYMS P04818 2/20 0.41
MAPK14 Q16539 1/20 0.41
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3710185 0.83 CYP2A6 (0.73) CYP2A6CYP1A2PAX8HPRT1CYP1B1
SCHEMBL476875 0.83 CYP2A6 (0.73) CYP2A6CYP1A2PAX8HPRT1CYP1B1
SCHEMBL9765602 0.82 CYP2A6 (0.67) CYP2A6CYP1A2PAX8HPRT1CA1
Hydrochloric Acid SCHEMBL8112381 0.81 CYP2A6 (0.70) CYP2A6CYP1A2PAX8HPRT1CYP1B1
SCHEMBL9644939 0.81 HPRT1 (0.70) CYP2A6CYP1A2PAX8HPRT1CA1
SCHEMBL5335748 0.80 CYP1A2 (0.43) CYP2A6CYP1A2CYP1A1CYP1B1NR4A2
SCHEMBL30186719 0.80 ALDH1A1 (0.65) CYP2A6CYP1A2PAX8HPRT1CA1
SCHEMBL268735 0.80 ALDH1A1 (0.65) CYP2A6CYP1A2PAX8HPRT1CA1
SCHEMBL29391827 0.80 ALDH1A1 (0.65) CYP2A6CYP1A2PAX8HPRT1CA1
SCHEMBL11723197 0.79 ALDH1A1 (0.48) CYP2A6CYP1A2PAX8CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0319073-B1 Cyclo-octane neuroprotective agents MERCK SHARP & DOHME (GB) 1995-08-23 EP disclosed
EP-0272621-B1 Method for the production of 5H-dibenzo[a,d]cyclohepten-5-ones BASF Aktiengesellschaft (DE) 1991-11-27 EP disclosed
US-4927819-A ANTICONVULSANT, PREVENTION OF NEURODEGENERATIVE DISORDERS MERCK SHARP & DOHME LIMITED (GB) 1990-05-22 US disclosed
US-4845302-A Preparation of 5H-dibenzo[a,d]cyclohepten-5-ones BASF AKTIENGSELLSCHAFT (DE) 1989-07-04 US disclosed
EP-0319073-A2 Cyclo-octane neuroprotective agents MERCK SHARP & DOHME LTD. (GB) 1989-06-07 EP disclosed
EP-0272621-A2 Method for the production of 5H-dibenzo[a,d]cyclohepten-5-ones BASF Aktiengesellschaft (DE) 1988-06-29 EP disclosed
EP-0115690-A1 Dibenzocycloheptenylidenes AMERICAN HOME PRODUCTS CORPORATION (US) 1984-08-15 EP disclosed
US-4003915-A ANTICONVULSANTS, PARKINSON*S DISEASE HOFFMANN-LA ROCHE INC. (US) 1977-01-18 US disclosed