SCHEMBL9212344

SCHEMBL9212344

CCOC(=O)C(=CN(C)C)C(=O)c1cc(F)c(F)c(Cl)c1F

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.40
CYP11B1 P15538 10/20 0.39
CYP11B2 P19099 8/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
MAPT P10636 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
GPR35 Q9HC97 2/20 0.36
GAA P10253 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9562415 1.00 CYP2C9 (0.40) CYP2C9CYP11B1CYP11B2MEN1KMT2A
SCHEMBL7519192 0.90 MEN1 (0.40) CYP2C9CYP11B1CYP11B2MEN1KMT2A
SCHEMBL7519196 0.90 MEN1 (0.40) CYP2C9CYP11B1CYP11B2MEN1KMT2A
SCHEMBL9561731 0.88 MEN1 (0.40) CYP2C9CYP11B1CYP11B2MEN1KMT2A
SCHEMBL4567521 0.88 MEN1 (0.40) CYP2C9CYP11B1CYP11B2MEN1KMT2A
SCHEMBL3695378 0.88 MEN1 (0.40) CYP2C9CYP11B1CYP11B2MEN1KMT2A
SCHEMBL30843044 0.88 MEN1 (0.40) CYP2C9CYP11B1CYP11B2MEN1KMT2A
SCHEMBL9486031 0.86 CYP11B1 (0.36) CYP2C9CYP11B1CYP11B2MEN1KMT2A
SCHEMBL9486024 0.86 CYP11B1 (0.36) CYP2C9CYP11B1CYP11B2MEN1KMT2A
SCHEMBL4887115 0.85 CES2 (0.49) CYP2C9CYP11B1CYP11B2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0457090-B1 Process for the preparation of 3-amino-2 (het)aroyl-acrylic acid derivatives BAYER AG (DE) 1995-11-29 EP disclosed
US-5182401-A Bactericide intermediate BAYER AKTIENGESELLSCHAFT (DE) 1993-01-26 US disclosed
EP-0457090-A2 Process for the preparation of 3-amino-2 (het)aroyl-acrylic acid derivatives BAYER AG (DE) 1991-11-21 EP disclosed