SCHEMBL9213658

SCHEMBL9213658

COc1ccc2c(CC(O)CN3CCC(CN4CCc5cc(C)c(C)cc5C4=O)C3)cccc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 3/20 0.41
RAD52 P43351 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
GAA P10253 3/20 0.41
PRMT5 O14744 2/20 0.40
WDR77 Q9BQA1 2/20 0.40
ADRB2 P07550 4/20 0.40
ADRB1 P08588 4/20 0.40
ADRB3 P13945 4/20 0.40
SIGMAR1 Q99720 1/20 0.39
MEN1 O00255 2/20 0.39
NTSR1 P30989 2/20 0.39
KMT2A Q03164 2/20 0.39
MAPT P10636 2/20 0.38
HTT P42858 2/20 0.38
IDH1 O75874 1/20 0.38
NPC1 O15118 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9211468 0.96 PRMT5 (0.41) ALDH1A1KDM4ERAD52NPSR1GAA
SCHEMBL9206642 0.95 PRMT5 (0.40) ALDH1A1KDM4ERAD52NPSR1GAA
Hydrochloric Acid SCHEMBL9212963 0.95 PRMT5 (0.40) ALDH1A1KDM4ERAD52NPSR1GAA
SCHEMBL9215245 0.93 ALDH1A1 (0.41) ALDH1A1KDM4ERAD52NPSR1GAA
SCHEMBL9206673 0.90 PRMT5 (0.38) ALDH1A1KDM4ERAD52NPSR1GAA
SCHEMBL9210433 0.88 PRMT5 (0.41) ALDH1A1KDM4ERAD52NPSR1GAA
Hydrochloric Acid SCHEMBL9215384 0.87 PRMT5 (0.40) ALDH1A1KDM4ERAD52NPSR1GAA
SCHEMBL9208294 0.86 PRMT5 (0.42) PRMT5WDR77
Hydrochloric Acid SCHEMBL9206928 0.86 PRMT5 (0.40) PRMT5WDR77
SCHEMBL9216938 0.85 PRMT5 (0.40) PRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed