SCHEMBL9213740

SCHEMBL9213740

COc1ccc2cc(CCN3CCC(CN4CCc5cc(C)c(C)cc5C4)C3)ccc2c1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.48
HTR1A P08908 4/20 0.47
SLC6A4 P31645 4/20 0.47
DHCR7 Q9UBM7 2/20 0.45
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9213303 0.94 MEN1 (0.49) ABCB1HTR1ASLC6A4DHCR7MEN1
Hydrochloric Acid SCHEMBL9216467 0.85 DHCR7 (0.58) ABCB1HTR1ASLC6A4DHCR7KMT2A
Hydrochloric Acid SCHEMBL9215875 0.84 ABCB1 (0.54) ABCB1HTR1ASLC6A4DHCR7
SCHEMBL9211025 0.83 HRH3 (0.49) ABCB1HTR1ASLC6A4MEN1KMT2A
SCHEMBL9215240 0.83 MEN1 (0.47) ABCB1HTR1ASLC6A4MEN1KMT2A
SCHEMBL9207036 0.82 HRH3 (0.50) ABCB1HTR1ASLC6A4MEN1KMT2A
SCHEMBL9211782 0.81 DHCR7 (0.51) ABCB1DHCR7
SCHEMBL9205910 0.81 DHCR7 (0.57) ABCB1DHCR7MEN1KMT2A
Hydrochloric Acid SCHEMBL9215735 0.80 ABCB1 (0.57) ABCB1SLC6A4MEN1KMT2A
Hydrochloric Acid SCHEMBL9206759 0.80 DHCR7 (0.64) ABCB1HTR1ASLC6A4DHCR7KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed