SCHEMBL9216836

SCHEMBL9216836

COc1ccc(OCCCN2CCC(CN3CCc4cc(OC)c(OC)cc4C3=O)C2)cc1

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.51
ADRA1B P35368 1/20 0.46
DRD2 P14416 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HTR1A P08908 1/20 0.43
DRD4 P21917 1/20 0.43
DRD3 P35462 1/20 0.43
TDP1 Q9NUW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9215591 0.99 ABCB1 (0.50) ABCB1ADRA1BDRD2MEN1KMT2A
SCHEMBL9206439 0.95 ABCB1 (0.49) ABCB1ADRA1BHTR1ADRD4DRD3
SCHEMBL9215106 0.94 ADRA1B (0.44) ABCB1ADRA1BDRD2
Hydrochloric Acid SCHEMBL9213140 0.94 ABCB1 (0.48) ABCB1ADRA1BHTR1ADRD4DRD3
SCHEMBL9740001 0.94 ADRA1B (0.45) ABCB1ADRA1BDRD2MEN1KMT2A
Hydrochloric Acid SCHEMBL9206636 0.93 ABCB1 (0.48) ABCB1ADRA1B
Hydrochloric Acid SCHEMBL9208133 0.90 TDP1 (0.44) ABCB1DRD2KMT2ADRD3TDP1
Hydrochloric Acid SCHEMBL9212198 0.88 ADRA1B (0.44) ADRA1BDRD2
Hydrochloric Acid SCHEMBL9211764 0.87 ADRA1B (0.43) ABCB1ADRA1BMEN1KMT2AHTR1A
Hydrochloric Acid SCHEMBL9209383 0.87 HRH3 (0.47) ADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed