SCHEMBL9219971

SCHEMBL9219971

COc1ccc(C[C@H](CS(=O)(=O)C(C)(C)C)C(=O)O)cc1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.56
PPARG P37231 2/20 0.49
KMT2A Q03164 1/20 0.48
PPARA Q07869 1/20 0.46
POLB P06746 2/20 0.44
CA2 P00918 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9444964 1.00 LDHA (0.56) LDHAPPARGKMT2APPARAPOLB
SCHEMBL9219968 1.00 LDHA (0.56) LDHAPPARGKMT2APPARAPOLB
SCHEMBL9226473 0.84 PPARA (0.48) PPARGKMT2APPARA
SCHEMBL9226476 0.84 PPARA (0.48) PPARGKMT2APPARA
SCHEMBL7269232 0.84 CYP1A2 (0.59)
SCHEMBL7163321 0.84 CYP1A2 (0.59)
SCHEMBL7277365 0.84 CYP1A2 (0.59)
SCHEMBL10436394 0.82 LDHA (0.76) LDHAPPARGKMT2APPARAPOLB
SCHEMBL8531043 0.80 CYP1A2 (0.42)
SCHEMBL12494157 0.79 LDHA (0.71) LDHAPPARGKMT2APPARAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5389616-A Renin inhibitor, hypotensive agent HOFFMAN-LAROCHE INC. (US) 1995-02-14 US disclosed
US-5256645-A Renin inhibitors; hypotensive agents HOFFMANN-LA ROCHE INC. (US) 1993-10-26 US disclosed
US-5134123-A Renin enzyme inhibitors for cardiovascular disorders and high blood pressure HOFFMAN-LA ROCHE INC. (US) 1992-07-28 US disclosed