SCHEMBL9220558

SCHEMBL9220558

CN(CCc1c[nH]c2nc(N)nc(O)c12)c1ccc(C(=O)N[C@@H](CCC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O)nc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYMS P04818 9/20 0.51
DHFR P00374 5/20 0.51
FPR2 P25090 3/20 0.44
FOLR1 P15328 7/20 0.43
SLC19A1 P41440 7/20 0.43
SLC46A1 Q96NT5 7/20 0.43
GART P22102 4/20 0.43
FOLR2 P14207 3/20 0.43
ATIC P31939 2/20 0.43
SHMT1 P34896 1/20 0.43
FRK P42685 1/20 0.43
KDM4E B2RXH2 1/20 0.42
TLR4 O00206 1/20 0.42
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
TP53 P04637 1/20 0.42
GLA P06280 1/20 0.42
POLB P06746 1/20 0.42
HMGB1 P09429 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9229379 1.00 TYMS (0.51) TYMSDHFRFPR2FOLR1SLC19A1
SCHEMBL9228615 0.89 DHFR (0.62) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL9228950 0.89 TYMS (0.49) TYMSDHFRFPR2FOLR1SLC19A1
SCHEMBL9223587 0.89 TYMS (0.49) TYMSDHFRFPR2FOLR1SLC19A1
SCHEMBL9220575 0.88 TYMS (0.44) TYMSDHFRFPR2FOLR1SLC19A1
SCHEMBL9555170 0.88 TYMS (0.50) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL9225400 0.86 DHFR (0.61) TYMSDHFRFPR2FOLR1SLC19A1
SCHEMBL9228560 0.86 DHFR (0.61) TYMSDHFRFPR2FOLR1SLC19A1
SCHEMBL9225966 0.86 TYMS (0.50) TYMSDHFRFOLR1SLC19A1SLC46A1
SCHEMBL9226053 0.86 TYMS (0.50) TYMSDHFRFOLR1SLC19A1SLC46A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5459129-A Antitumor agents; enzyme inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-10-17 US disclosed
US-5268362-A Containing benzene and purine rings TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-12-07 US disclosed
EP-0492316-A1 Condensed heterocyclic oligoglutamate derivatives, their production and pharmaceutical compositions containing them Takeda Chemical Industries, Ltd. (JP) 1992-07-01 EP disclosed