SCHEMBL9220601

SCHEMBL9220601

CNCC1CSc2ccc(F)cc2C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 1/20 0.39
SLC6A4 P31645 10/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
HTR2B P41595 4/20 0.35
HTR2A P28223 2/20 0.35
HTR2C P28335 1/20 0.35
SLC6A2 P23975 9/20 0.34
SLC6A3 Q01959 6/20 0.34
AQP1 P29972 2/20 0.33
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
CYP2D6 P10635 3/20 0.32
CYP2C19 P33261 3/20 0.32
KCNH2 Q12809 2/20 0.32
CYP3A4 P08684 1/20 0.32
CDK4 P11802 1/20 0.32
PRKACA P17612 1/20 0.32
PRKACG P22612 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9209494 0.80 MALT1 (0.38) MALT1SLC6A4ADRA2AADRA2BADRA2C
SCHEMBL9215221 0.80 MALT1 (0.36) MALT1SLC6A4ADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL9273659 0.78 HTR2A (0.37) MALT1SLC6A4ADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL9278206 0.77 MALT1 (0.35) MALT1SLC6A4ADRA2AADRA2BADRA2C
SCHEMBL9210918 0.75 MALT1 (0.43) MALT1HTR2BHTR2C
SCHEMBL9869729 0.74 MALT1 (0.38) MALT1
Hydrochloric Acid SCHEMBL9274817 0.73 DRD2 (0.38) SLC6A4ADRA2CHTR2BHTR2AHTR2C
Hydrochloric Acid SCHEMBL9275494 0.72 KDM4E (0.38) SLC6A4ADRA2CHTR2BHTR2AHTR2C
SCHEMBL9220092 0.71 DRD2 (0.46) SLC6A4HTR2BHTR2AHTR2CSLC6A3
SCHEMBL9210567 0.70 HTR2A (0.40) HTR2BHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0389425-B1 Benzotiopyranyl amines CIBA GEIGY AG (CH) 1995-04-26 EP disclosed
US-5071858-A Antipsychotic benzothiopyranylamines CIBA-GEIGY CORPORATION (US) 1991-12-10 US disclosed
EP-0389425-A1 Benzotiopyranyl amines CIBA-GEIGY AG (CH) 1990-09-26 EP disclosed