SCHEMBL9220965

SCHEMBL9220965

Cc1cc(C)c(NC(=O)N(Cc2ccc3c(c2)=c2ccccc2=3)C2CCCCCC2)c(C)c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
UBE2M P61081 8/20 0.43
DCUN1D1 Q96GG9 8/20 0.43
TP53 P04637 4/20 0.43
MAPT P10636 1/20 0.43
ALDH1A1 P00352 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 3/20 0.42
THRB P10828 1/20 0.41
KDM4E B2RXH2 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9220959 0.88 GAA (0.50) GAANPSR1UBE2MDCUN1D1TP53
SCHEMBL8808845 0.87 GAA (0.51) GAANPSR1UBE2MDCUN1D1TP53
SCHEMBL9056936 0.86 GAA (0.50) GAANPSR1UBE2MDCUN1D1TP53
SCHEMBL9059369 0.85 GAA (0.49) GAANPSR1UBE2MDCUN1D1TP53
SCHEMBL9220408 0.85 GAA (0.47) GAANPSR1UBE2MDCUN1D1TP53
SCHEMBL8809220 0.84 NPSR1 (0.48) GAANPSR1UBE2MDCUN1D1TP53
SCHEMBL8809108 0.84 GAA (0.48) GAANPSR1UBE2MDCUN1D1TP53
SCHEMBL8807120 0.84 GAA (0.48) GAANPSR1UBE2MDCUN1D1TP53
SCHEMBL8811763 0.84 GCGR (0.47) GAANPSR1UBE2MDCUN1D1TP53
SCHEMBL8809779 0.84 GAA (0.52) GAANPSR1UBE2MDCUN1D1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5420348-A Enzyme inhibitors YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
EP-0447116-B1 Urea derivatives, their production, and pharmaceutical compositions containing them YAMANOUCHI PHARMA CO LTD (JP) 1994-12-14 EP disclosed
US-5258405-A Acetyl coenzyme A cholesterol acetyltransferase inhibitors for cardiovascular disorders and atherosclerosis and antilipemic agents YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1993-11-02 US disclosed
EP-0447116-A1 Urea derivatives, their production, and pharmaceutical compositions containing them YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1991-09-18 EP disclosed