SCHEMBL9225829

SCHEMBL9225829

Nc1nc(O)c2c(CCc3ccc(C(=O)N[C@@H](CCC(=O)N[C@@H](CCC(=O)O)C(=O)O)C(=O)O)s3)c[nH]c2n1

nearest known ligand 0.70

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FOLR1 P15328 12/20 0.70
SLC46A1 Q96NT5 9/20 0.70
SLC19A1 P41440 6/20 0.70
GART P22102 11/20 0.63
DHFR P00374 3/20 0.56
TYMS P04818 3/20 0.56
ATIC P31939 6/20 0.50
FOLR2 P14207 5/20 0.50
SHMT1 P34896 4/20 0.49
FRK P42685 1/20 0.49
SHMT2 P34897 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9224206 1.00 FOLR1 (0.70) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9439839 0.97 FOLR1 (0.74) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9221924 0.92 FOLR1 (0.71) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9228411 0.92 FOLR1 (0.71) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9439673 0.92 FOLR1 (0.75) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9227773 0.91 FOLR1 (0.66) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9223823 0.91 FOLR1 (0.66) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9439748 0.89 FOLR1 (0.75) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9439759 0.89 FOLR1 (0.75) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9564163 0.89 FOLR1 (0.62) FOLR1SLC46A1SLC19A1GARTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0492316-A1 Condensed heterocyclic oligoglutamate derivatives, their production and pharmaceutical compositions containing them Takeda Chemical Industries, Ltd. (JP) 1992-07-01 EP claimed
US-5459129-A Antitumor agents; enzyme inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-10-17 US disclosed
US-5268362-A Containing benzene and purine rings TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-12-07 US disclosed
EP-0492316-A1 Condensed heterocyclic oligoglutamate derivatives, their production and pharmaceutical compositions containing them Takeda Chemical Industries, Ltd. (JP) 1992-07-01 EP disclosed