SCHEMBL9439673

SCHEMBL9439673

Nc1nc(O)c2c(CCCc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)s3)c[nH]c2n1

nearest known ligand 0.75

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FOLR1 P15328 13/20 0.75
SLC46A1 Q96NT5 9/20 0.75
SLC19A1 P41440 6/20 0.75
GART P22102 11/20 0.72
DHFR P00374 3/20 0.56
TYMS P04818 3/20 0.56
FOLR2 P14207 6/20 0.55
ATIC P31939 6/20 0.55
SHMT1 P34896 4/20 0.51
SHMT2 P34897 3/20 0.51
FRK P42685 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9439839 0.95 FOLR1 (0.74) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9439728 0.92 FOLR1 (0.76) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9225829 0.92 FOLR1 (0.70) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9224206 0.92 FOLR1 (0.70) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9439758 0.90 FOLR1 (0.76) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9564163 0.90 FOLR1 (0.62) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9221180 0.89 FOLR1 (0.71) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9439922 0.87 FOLR1 (0.57) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9439748 0.87 FOLR1 (0.75) FOLR1SLC46A1SLC19A1GARTDHFR
SCHEMBL9439759 0.87 FOLR1 (0.75) FOLR1SLC46A1SLC19A1GARTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3173890-A None JP disclosed
US-5354754-A Antitumor and -carcinogenic agents; treating human epidermoid carcinoma KB TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-10-11 US disclosed
JP-H03173890-A PYRROLO(2,3-D)PYRIMIDINE DERIVATIVE, ITS PRODUCTION, USE AND INTERMEDIATE TAKEDA CHEM IND LTD 1991-07-29 JP disclosed
EP-0418924-A2 Pyrrolopyrimidines, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-03-27 EP disclosed