SCHEMBL9227129

SCHEMBL9227129

Nc1nc(O)c2c(CCc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)C(C[C@H](N)C(=O)O)C(=O)O)cc3)c[nH]c2n1

nearest known ligand 0.67

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DHFR P00374 12/20 0.67
TYMS P04818 6/20 0.67
FOLR1 P15328 2/20 0.59
SLC19A1 P41440 2/20 0.59
SLC46A1 Q96NT5 2/20 0.59
GART P22102 2/20 0.59
ATIC P31939 2/20 0.59
FOLR2 P14207 1/20 0.59
SHMT1 P34896 1/20 0.59
FRK P42685 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9223626 0.95 DHFR (0.61) DHFRTYMSFOLR1SLC19A1SLC46A1
SCHEMBL9555370 0.93 DHFR (0.68) DHFRTYMSFOLR1SLC19A1SLC46A1
SCHEMBL9691063 0.91 DHFR (0.62) DHFRTYMSFOLR1SLC19A1SLC46A1
SCHEMBL9221717 0.90 DHFR (0.54) DHFRTYMSFOLR1SLC19A1SLC46A1
SCHEMBL9225411 0.89 DHFR (0.53) DHFRTYMSFOLR1SLC19A1SLC46A1
SCHEMBL9227909 0.89 DHFR (0.53) DHFRTYMSFOLR1SLC19A1SLC46A1
SCHEMBL9223738 0.89 DHFR (0.53) DHFRTYMSFOLR1SLC19A1SLC46A1
Pemetrexed SCHEMBL7848273 0.89 DHFR (0.83) DHFRTYMSFOLR1SLC19A1SLC46A1
Pemetrexed SCHEMBL12022769 0.89 DHFR (0.83) DHFRTYMSFOLR1SLC19A1SLC46A1
SCHEMBL9223819 0.88 DHFR (0.62) DHFRTYMSFOLR1SLC19A1SLC46A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5268362-A Containing benzene and purine rings TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-12-07 US claimed
EP-0492316-A1 Condensed heterocyclic oligoglutamate derivatives, their production and pharmaceutical compositions containing them Takeda Chemical Industries, Ltd. (JP) 1992-07-01 EP claimed
US-5459129-A Antitumor agents; enzyme inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-10-17 US disclosed
US-5268362-A Containing benzene and purine rings TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-12-07 US disclosed
EP-0492316-A1 Condensed heterocyclic oligoglutamate derivatives, their production and pharmaceutical compositions containing them Takeda Chemical Industries, Ltd. (JP) 1992-07-01 EP disclosed