SCHEMBL9230342

SCHEMBL9230342

CC(C)N1C[C@@H](COS(C)(=O)=O)OC1=O

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 1/20 0.41
MAOA P21397 1/20 0.35
GRM2 Q14416 5/20 0.34
MAPK1 P28482 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9230346 1.00 HTR2B (0.41) HTR2BMAOAGRM2MAPK1L3MBTL1
SCHEMBL8659488 0.82 HTR2B (0.37) HTR2B
SCHEMBL14168007 0.82 HTR2B (0.46) HTR2BGRM2MAPK1L3MBTL1
SCHEMBL7911772 0.81 HTR2B (0.50) HTR2BMAOAGRM2MAPK1L3MBTL1
SCHEMBL15247384 0.80 PTPN1 (0.37) GRM2MAPK1L3MBTL1
SCHEMBL4921609 0.80 CYP2D6 (0.47) HTR2BGRM2MAPK1
SCHEMBL4953038 0.80 CYP2D6 (0.47) HTR2BGRM2MAPK1
SCHEMBL14168364 0.80 MAOA (0.38) MAOAGRM2MAPK1L3MBTL1
SCHEMBL10151437 0.80 MAOA (0.38) MAOAGRM2MAPK1L3MBTL1
SCHEMBL14173675 0.78 HTR2B (0.40) HTR2BMAOAGRM2MAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647634-A1 Method of preparing a heterocyclic intermediate for the production of optically active aryloxy-substituted vicinal aminoalcohols DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1995-04-12 EP disclosed
EP-0647633-A1 Method of preparing a heterocyclic intermediate for the production of optically active aryloxysubstituted vicinal aminoalcohols DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1995-04-12 EP disclosed
EP-0153746-B1 3-AMINO-2-HYDROXYPROPYL DERIVATIVES OF PYRIMIDIN-4-ONE MERCK & CO. INC. (US) 1990-11-22 EP disclosed
US-4602093-A ADRENERGIC BLOCKING AGENTS MERCK & CO., INC. (US) 1986-07-22 US disclosed
US-4598149-A ADRENERGIC BLOCKING AGENTS MERCK & CO., INC. (US) 1986-07-01 US disclosed
EP-0153746-A2 3-Amino-2-hydroxypropyl derivatives of pyrimidin-4-one MERCK & CO. INC. (US) 1985-09-04 EP disclosed