SCHEMBL9230477

SCHEMBL9230477

COc1ccc2c(c1)C(CO)(N(C)C)CCO2

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
APP P05067 2/20 0.41
BACE1 P56817 2/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
CYP3A4 P08684 1/20 0.37
CTNNB1 P35222 1/20 0.36
WNT3A P56704 1/20 0.36
SIGMAR1 Q99720 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9232640 0.81 MAP3K14 (0.48) APPBACE1
Hydrochloric Acid SCHEMBL9234205 0.81 BACE1 (0.39) APPBACE1CTNNB1WNT3AKCNH2
SCHEMBL9233832 0.81 AKR1B1 (0.51) APPBACE1CTNNB1
Hydrochloric Acid SCHEMBL9233886 0.76 KMT2A (0.36) KMT2ASMN1; SMN2
Hydrochloric Acid SCHEMBL9228764 0.75 MAPT (0.41) MEN1KMT2ACYP2C9CYP3A4SMN1; SMN2
Hydrochloric Acid SCHEMBL9232618 0.75 APP (0.38) APPBACE1CYP3A4SMN1; SMN2
SCHEMBL9228772 0.73 RYR2 (0.39) CYP2C9TSHRCYP2C19CYP3A4KCNH2
SCHEMBL6580916 0.71 RAB9A (0.43) APPBACE1MEN1KMT2ATSHR
SCHEMBL6578320 0.70 SMN1; SMN2 (0.42) APPBACE1MEN1KMT2ATSHR
SCHEMBL8793923 0.70 AKR1B1 (0.46) BACE1MEN1KMT2ATSHRCTNNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0639557-A1 TRIALKYLAMINE DERIVATIVE AND AMELIORANT FOR DIGESTIVE TRACT MOVEMENT CONTAINING THE SAME ZERIA PHARMACEUTICAL CO., LTD. (JP) 1995-02-22 EP disclosed
US-5380748-A Trialkylamine derivative and ameliorant for digestive tract movement containing the same ZERIA PHARMACEUTICAL CO., LTD. (JP) 1995-01-10 US disclosed