SCHEMBL9230683

SCHEMBL9230683

CN(C)c1cc(NC(=O)C2CCC(CN)CC2)ccn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 7/20 0.45
ACVRL1 P37023 2/20 0.44
F11 P03951 4/20 0.44
KLKB1 P03952 1/20 0.43
PRSS1 P07477 1/20 0.43
PRSS2 P07478 1/20 0.43
PRSS3 P35030 1/20 0.43
ROCK2 O75116 4/20 0.43
ROCK1 Q13464 4/20 0.43
PKN2 Q16513 3/20 0.43
RPS6KA5 O75582 2/20 0.43
LRRK2 Q5S007 2/20 0.43
TP53 P04637 2/20 0.43
CYP3A4 P08684 2/20 0.43
MAPK14 Q16539 1/20 0.43
CHUK O15111 1/20 0.43
PRKD3 O94806 1/20 0.43
CDK1 P06493 1/20 0.43
CDK2 P24941 1/20 0.43
LTK P29376 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9230680 1.00 TYK2 (0.45) TYK2ACVRL1F11KLKB1PRSS1
SCHEMBL1553681 0.84 SMARCA2 (0.49) TYK2ACVRL1F11KLKB1PRSS1
SCHEMBL1553679 0.84 SMARCA2 (0.49) TYK2ACVRL1F11KLKB1PRSS1
SCHEMBL9229123 0.84 ACVRL1 (0.51) TYK2ACVRL1JAK2JAK1CDK9
SCHEMBL9229125 0.84 ACVRL1 (0.51) TYK2ACVRL1JAK2JAK1CDK9
SCHEMBL1552890 0.83 ABL1 (0.49) TYK2ACVRL1F11KLKB1PRSS1
SCHEMBL1552889 0.83 ABL1 (0.49) TYK2ACVRL1F11KLKB1PRSS1
SCHEMBL9231780 0.82 ACVRL1 (0.54) TYK2ACVRL1JAK2JAK1CDK9
SCHEMBL9231785 0.82 ACVRL1 (0.54) TYK2ACVRL1JAK2JAK1CDK9
SCHEMBL9234289 0.81 TYK2 (0.59) TYK2ACVRL1JAK2JAK1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5478838-A Treating hypertension, angina pectoris, asthma, improving peripheral circulation YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-12-26 US disclosed
EP-0641781-A1 4-AMINO(ALKYL)CYCLOHEXANE-1-CARBOXAMIDE COMPOUND AND USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-03-08 EP disclosed