SCHEMBL9236325

SCHEMBL9236325

Cc1ccc(C[C@@H]2CN(CCNC(=O)c3cccnc3)CCN2C(=O)c2cc(C(F)(F)F)cc(C(F)(F)F)c2)cc1C

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
TACR1 P25103 7/20 0.41
NAMPT P43490 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
CSF1R P07333 1/20 0.39
BRAF P15056 1/20 0.39
TRPA1 O75762 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8836811 1.00 ADRA2A (0.44) ADRA2AADRA2BADRA2CTACR1NAMPT
SCHEMBL8836478 0.96 SMN1; SMN2 (0.44) ADRA2AADRA2BADRA2CTACR1NAMPT
SCHEMBL7830364 0.96 SMN1; SMN2 (0.44) ADRA2AADRA2BADRA2CTACR1NAMPT
Hydrochloric Acid SCHEMBL7560436 0.87 TACR1 (0.42) TACR1
Hydrochloric Acid SCHEMBL8476084 0.86 TACR1 (0.44) TACR1
Hydrochloric Acid SCHEMBL9233950 0.86 TACR1 (0.44) TACR1
Hydrochloric Acid SCHEMBL9241357 0.85 TACR1 (0.48) TACR1
Hydrochloric Acid SCHEMBL7556699 0.85 TACR1 (0.42) TACR1
Hydrochloric Acid SCHEMBL7560528 0.85 TACR1 (0.41) TACR1
Hydrochloric Acid SCHEMBL8480146 0.84 TACR1 (0.43) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0655442-A1 Piperazine derivatives as Tachykinin antagonists FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1995-05-31 EP disclosed