SCHEMBL9237132

SCHEMBL9237132

[CH2]CCC=Cc1ccc2sccc2c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.53
DYRK1A Q13627 1/20 0.35
CA2 P00918 5/20 0.34
MRGPRX4 Q96LA9 2/20 0.34
CTNNB1 P35222 1/20 0.34
WNT3A P56704 1/20 0.34
CA12 O43570 4/20 0.33
PTPRC P08575 1/20 0.32
PTPN6 P29350 1/20 0.32
PTPN11 Q06124 1/20 0.32
PTPN22 Q9Y2R2 1/20 0.32
DRD2 P14416 1/20 0.31
DRD3 P35462 1/20 0.31
KCNH2 Q12809 1/20 0.31
HDAC1 Q13547 1/20 0.30
HDAC8 Q9BY41 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9432076 0.80 CYP2A6 (0.70) CYP2A6DYRK1ACA2MRGPRX4CTNNB1
SCHEMBL6958280 0.80 CYP2A6 (0.56) CYP2A6DYRK1ACA2MRGPRX4CTNNB1
SCHEMBL6958287 0.80 CYP2A6 (0.56) CYP2A6DYRK1ACA2MRGPRX4CTNNB1
SCHEMBL9111250 0.78 CYP2A6 (0.36) CYP2A6MRGPRX4HDAC1HDAC8
SCHEMBL9111666 0.75 CYP2A6 (0.58) CYP2A6DYRK1ACA2MRGPRX4CTNNB1
SCHEMBL13177010 0.73 CYP2A6 (0.66) CYP2A6DYRK1ACA2CTNNB1WNT3A
SCHEMBL9819834 0.73 RELA (0.55) KCNH2HDAC1HDAC8
SCHEMBL8735739 0.73 RELA (0.55) KCNH2HDAC1HDAC8
SCHEMBL21457945 0.70 CYP2A6 (0.56) CYP2A6DYRK1ACA2MRGPRX4CTNNB1
SCHEMBL21457942 0.70 CYP2A6 (0.56) CYP2A6DYRK1ACA2CTNNB1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0670831-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-09-13 EP disclosed
WO-1995009159-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1995-04-06 WO disclosed