SCHEMBL9239106

SCHEMBL9239106

COc1ccc2c(c1)-c1c(ccn1CCN)C2

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 11/20 0.69
HTR2A P28223 11/20 0.69
DRD2 P14416 4/20 0.42
DRD1 P21728 4/20 0.42
DRD5 P21918 4/20 0.42
DRD3 P35462 4/20 0.42
METAP1 P53582 1/20 0.40
DRD4 P21917 2/20 0.39
GAA P10253 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ACHE P22303 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8873552 0.90 HTR2C (0.57) HTR2CHTR2ADRD2DRD1DRD5
Fumaric Acid SCHEMBL8873545 0.90 HTR2C (0.57) HTR2CHTR2ADRD2DRD1DRD5
SCHEMBL8875204 0.89 HTR2C (0.55) HTR2CHTR2ADRD2DRD1DRD5
SCHEMBL8596870 0.88 HTR2C (0.67) HTR2CHTR2ADRD2DRD1DRD5
SCHEMBL8599014 0.82 HTR2C (1.00) HTR2CHTR2AMETAP1
SCHEMBL8595428 0.82 HTR2C (1.00) HTR2CHTR2AMETAP1
SCHEMBL8595714 0.82 HTR2C (1.00) HTR2CHTR2AMETAP1
SCHEMBL9238901 0.81 HTR2A (0.55) HTR2CHTR2ADRD2DRD1DRD5
SCHEMBL8596868 0.81 HTR2C (0.65) HTR2CHTR2ADRD2DRD1DRD5
Fumaric Acid SCHEMBL8875270 0.80 HTR2A (0.47) HTR2CHTR2AGAAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0657426-A2 Tricyclic pyrrole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-06-14 EP disclosed