SCHEMBL9240100

SCHEMBL9240100

CC(C)(C)n1ncc(SCc2ccc(C(F)(F)F)cc2)c(Cl)c1=O

nearest known ligand 0.82

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.82
RAB9A P51151 2/20 0.82
MEN1 O00255 1/20 0.82
GALR3 O60755 1/20 0.82
NR2F2 P24468 1/20 0.82
GPR183 P32249 1/20 0.82
KMT2A Q03164 1/20 0.82
GPR35 Q9HC97 1/20 0.82
MAPT P10636 3/20 0.51
GAA P10253 2/20 0.51
PKM P14618 1/20 0.51
LMNA P02545 5/20 0.41
TOP2A P11388 1/20 0.41
NPBWR1 P48145 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
EGLN1 Q9GZT9 1/20 0.39
HTT P42858 3/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9775203 0.94 NPC1 (0.72) NPC1RAB9AMEN1GALR3NR2F2
Pyridaben SCHEMBL27429 0.90 MEN1 (1.00) NPC1RAB9AMEN1GALR3NR2F2
Pyridaben SCHEMBL8372466 0.90 MEN1 (1.00) NPC1RAB9AMEN1GALR3NR2F2
SCHEMBL9775193 0.88 NPC1 (0.81) NPC1RAB9AMEN1GALR3NR2F2
SCHEMBL9775172 0.87 MEN1 (0.76) NPC1RAB9AMEN1GALR3NR2F2
SCHEMBL9238518 0.86 MEN1 (0.76) NPC1RAB9AMEN1GALR3NR2F2
SCHEMBL29458630 0.85 NPC1 (0.77) NPC1RAB9AMEN1GALR3NR2F2
SCHEMBL9234574 0.85 RAB9A (0.77) NPC1RAB9AMEN1GALR3NR2F2
SCHEMBL9775168 0.83 MEN1 (0.74) NPC1RAB9AMEN1GALR3NR2F2
SCHEMBL9238805 0.83 MEN1 (0.74) NPC1RAB9AMEN1GALR3NR2F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0665223-A1 Antitumor agent, novel 3(2H)-pyridazinone derivatives and their preparation TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-08-02 EP disclosed