SCHEMBL9241237

SCHEMBL9241237

CCCC1COC(C#Cc2ccc(-c3ccc(F)c(F)c3)nc2)OC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.38
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
PKM P14618 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
GRM5 P41594 3/20 0.32
NSD2 O96028 1/20 0.32
KDM1A O60341 3/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
HTT P42858 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
RPS6KB1 P23443 1/20 0.30
AKT1 P31749 1/20 0.30
PDE5A O76074 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9241228 1.00 GRM2 (0.38) GRM2NPC1TP53PKMRAB9A
SCHEMBL9246721 0.94 GRM2 (0.37) GRM2NPC1TP53PKMRAB9A
SCHEMBL9250105 0.94 GRM2 (0.37) GRM2NPC1TP53PKMRAB9A
SCHEMBL9247841 0.93 GRM2 (0.37) GRM2NPC1TP53PKMRAB9A
SCHEMBL9247847 0.93 GRM2 (0.37) GRM2NPC1TP53PKMRAB9A
SCHEMBL9246509 0.91 GRM2 (0.33) GRM2NPC1TP53PKMRAB9A
SCHEMBL9246504 0.91 GRM2 (0.33) GRM2NPC1TP53PKMRAB9A
SCHEMBL9243964 0.88 GRM5 (0.43) NPC1RAB9ASMN1; SMN2CYP11B1CYP11B2
SCHEMBL9243972 0.88 GRM5 (0.43) NPC1RAB9ASMN1; SMN2CYP11B1CYP11B2
SCHEMBL9246705 0.87 NPY5R (0.31) GRM2KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5447657-A Liquid crystal compounds HOFFMANN-LA ROCHE INC. (US) 1995-09-05 US claimed
US-5447657-A Liquid crystal compounds HOFFMANN-LA ROCHE INC. (US) 1995-09-05 US disclosed