SCHEMBL9244385

SCHEMBL9244385

CCNCC1CCN(c2c(C(=O)O)c(=O)c3cc(F)cc(F)c3n2C2CC2)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.41
PIM1 P11309 2/20 0.37
GSK3A P49840 2/20 0.37
GSK3B P49841 2/20 0.37
PIM3 Q86V86 2/20 0.37
CSNK1G1 Q9HCP0 1/20 0.37
TOP1 P11387 2/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
KDM4E B2RXH2 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
CYP1A2 P05177 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9249913 0.92 KCNH2 (0.41) KCNH2PIM1GSK3AGSK3BPIM3
SCHEMBL9634933 0.79 PIM1 (0.38) KCNH2PIM1GSK3AGSK3BPIM3
SCHEMBL10730540 0.78 KCNH2 (0.52) KCNH2PIM1GSK3AGSK3BPIM3
SCHEMBL9129061 0.76 PIM1 (0.37) KCNH2PIM1GSK3AGSK3BPIM3
SCHEMBL9129070 0.76 PIM1 (0.37) KCNH2PIM1GSK3AGSK3BPIM3
SCHEMBL9215466 0.74 KDM4E (0.33) KCNH2PIM1GSK3AGSK3BPIM3
Pd-117558 SCHEMBL8922444 0.73 KCNH2 (0.65) KCNH2ALDH1A1POLBCHRM2CHRM1
Pd-117558 SCHEMBL10529381 0.73 KCNH2 (0.64) KCNH2ALDH1A1POLBCHRM2CHRM1
SCHEMBL10574861 0.72 KCNH2 (0.70) KCNH2ALDH1A1POLBCHRM2CHRM1
SCHEMBL9457173 0.72 KCNH2 (0.42) KCNH2PIM1GSK3AGSK3BPIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5476950-A Aminopyrrolidine compound DAIICHI SEIYAKU CO., LTD. (JP) 1995-12-19 US disclosed
US-5416222-A Chemical intermediates to prepare pyridinocarboxylic acid derivatives with high antimicrobial activity and excellent pharmacokinetics DAIICHI SEIYAKU CO., LTD. (JP) 1995-05-16 US disclosed
US-5380874-A Pyrrolidine carbamates DAIICHI SEIYAKU CO., LTD. (JP) 1995-01-10 US disclosed
US-5098912-A Bactericides for grampositive bacteria DAIICHI SEIYAKU CO., LTD. (JP) 1992-03-24 US disclosed