SCHEMBL9247451

SCHEMBL9247451

CC=CC1CCC(C#Cc2ccc(-c3ccc(F)c(F)c3)nc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.37
PTGES O14684 2/20 0.36
GRM5 P41594 1/20 0.33
BACE1 P56817 3/20 0.33
BACE2 Q9Y5Z0 1/20 0.33
CYP11B1 P15538 1/20 0.33
CYP11B2 P19099 1/20 0.33
NSD2 O96028 1/20 0.33
KDM1A O60341 2/20 0.32
EGLN1 Q9GZT9 1/20 0.32
CTSD P07339 1/20 0.31
NPC1 O15118 1/20 0.31
TP53 P04637 1/20 0.31
PKM P14618 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B10 Q99714 1/20 0.31
KMO O15229 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9247442 1.00 GRM2 (0.37) GRM2PTGESGRM5BACE1BACE2
SCHEMBL9247454 1.00 GRM2 (0.37) GRM2PTGESGRM5BACE1BACE2
SCHEMBL9247447 1.00 GRM2 (0.37) GRM2PTGESGRM5BACE1BACE2
SCHEMBL9244993 0.91 PTGES (0.36) GRM2PTGESGRM5BACE1BACE2
SCHEMBL9244982 0.91 PTGES (0.36) GRM2PTGESGRM5BACE1BACE2
SCHEMBL9244989 0.91 PTGES (0.36) GRM2PTGESGRM5BACE1BACE2
SCHEMBL9244978 0.91 PTGES (0.36) GRM2PTGESGRM5BACE1BACE2
SCHEMBL9246651 0.89 GRM2 (0.38) GRM2PTGESGRM5BACE1BACE2
SCHEMBL9246662 0.89 GRM2 (0.38) GRM2PTGESGRM5BACE1BACE2
SCHEMBL9246666 0.89 GRM2 (0.38) GRM2PTGESGRM5BACE1BACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5447657-A Liquid crystal compounds HOFFMANN-LA ROCHE INC. (US) 1995-09-05 US disclosed