SCHEMBL9251195

SCHEMBL9251195

O=C1NC(=S)SC1=Cc1cccc(Cl)c1Cl

nearest known ligand 0.78

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 3/20 0.78
CRHBP P24387 2/20 0.62
CRHR2 Q13324 2/20 0.62
PTP4A3 O75365 1/20 0.62
NAT1 P18440 7/20 0.61
MYC P01106 2/20 0.57
MAX P61244 2/20 0.57
CISD1 Q9NZ45 1/20 0.57
PDE4B Q07343 1/20 0.56
GSK3B P49841 1/20 0.56
PLA2G1B P04054 1/20 0.56
ATG4B Q9Y4P1 1/20 0.56
CA2 P00918 1/20 0.55
EPHX1 P07099 1/20 0.55
INSR P06213 1/20 0.54
IGF1R P08069 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9251192 1.00 PIM1 (0.78) PIM1CRHBPCRHR2PTP4A3NAT1
SCHEMBL12892060 0.88 PIM1 (1.00) PIM1CRHBPCRHR2PTP4A3NAT1
SCHEMBL13499561 0.86 PIM1 (0.74) PIM1CRHBPCRHR2PTP4A3NAT1
SCHEMBL18103052 0.86 PIM1 (0.74) PIM1CRHBPCRHR2PTP4A3NAT1
SCHEMBL18102944 0.86 PIM1 (0.74) PIM1CRHBPCRHR2PTP4A3NAT1
SCHEMBL1247443 0.85 PIM1 (0.62) PIM1NAT1IGF1R
SCHEMBL1247444 0.85 PIM1 (0.62) PIM1NAT1IGF1R
SCHEMBL14661291 0.83 PIM1 (0.70) PIM1CRHBPCRHR2PTP4A3NAT1
SCHEMBL13499565 0.83 PIM1 (0.70) PIM1CRHBPCRHR2PTP4A3NAT1
SCHEMBL14661290 0.83 PIM1 (0.70) PIM1CRHBPCRHR2PTP4A3NAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5464856-A Arylmethylenyl derivatives of imidazolidinones useful as antiinflammatory agents WARNER-LAMBERT COMPANY (US) 1995-11-07 US disclosed
US-5306822-A Mono-, di- or tri-methoxyphenylmethylene-2-thioxo-4-oxazolidinone as antihistamines WARNER-LAMBERT COMPANY (US) 1994-04-26 US disclosed
US-5208250-A Known and selected novel arylmethylenyl derivatives of thiazolidinones, imidazolidinones and oxazolidinones useful as antiallergy agents and anti-inflammatory agents WARNER-LAMBERT COMPANY (US) 1993-05-04 US disclosed
EP-0343643-A2 Arylmethylenyl derivatives of thiazolidnones, imidazolidinones and oxazolidinones useful as antiallergy agents and antiinflamatory agents WARNER-LAMBERT COMPANY (US) 1989-11-29 EP disclosed