SCHEMBL9252099

SCHEMBL9252099

O=C1c2ccccc2C(=O)N1Cc1cncs1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.47
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 1/20 0.46
PKM P14618 1/20 0.46
KMT2A Q03164 1/20 0.46
MAPK1 P28482 1/20 0.45
TSHR P16473 1/20 0.44
MAPT P10636 3/20 0.44
RECQL P46063 1/20 0.44
CASP3 P42574 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.42
SLC6A3 Q01959 1/20 0.42
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.41
HPGD P15428 1/20 0.41
XIAP P98170 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9933687 0.83 HDAC4 (0.41) GRM5ALDH1A1MEN1KMT2AMAPK1
SCHEMBL7666711 0.75 MAPK1 (0.56) ALDH1A1MEN1PKMKMT2AMAPK1
SCHEMBL1619449 0.74 ALDH1A1 (0.68) ALDH1A1MEN1PKMKMT2ATSHR
SCHEMBL25238058 0.72 MAPK1 (0.56) ALDH1A1MEN1PKMKMT2AMAPK1
SCHEMBL31202611 0.72 MAPK1 (0.56) ALDH1A1MEN1PKMKMT2AMAPK1
SCHEMBL5653134 0.71 MAPK1 (0.55) ALDH1A1MEN1PKMKMT2AMAPK1
SCHEMBL4651618 0.71 MAPK1 (0.59) ALDH1A1MEN1PKMKMT2AMAPK1
SCHEMBL8217760 0.70 POLB (0.48) GRM5ALDH1A1MEN1PKMKMT2A
SCHEMBL8052946 0.70 MEN1 (0.40) GRM5ALDH1A1MEN1PKMKMT2A
SCHEMBL7503789 0.70 MAPK1 (0.43) ALDH1A1MEN1PKMKMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5395838-A Aromatic aminomethyl substitutes compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-03-07 US disclosed
EP-0373891-B1 Anti-tumour agents ICI PLC (GB) 1994-11-02 EP disclosed
US-5252573-A Quinazoline derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-10-12 US disclosed
US-5089499-A Anticarcinogenic agents; thymidylate synthetase inhibitors; antiallergens; psoriasis IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-02-18 US disclosed
EP-0373891-A2 Anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-06-20 EP disclosed