SCHEMBL9255224

SCHEMBL9255224

COC(=O)CCNC(=O)c1ccc2c(c1)nc(-c1ccc(C#N)cc1)n2Cc1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.46
JAK2 O60674 1/20 0.45
JAK1 P23458 1/20 0.45
TYK2 P29597 1/20 0.45
JAK3 P52333 1/20 0.45
PTGER4 P35408 3/20 0.44
AR P10275 1/20 0.44
ADORA2A P29274 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
NAMPT P43490 5/20 0.41
ITK Q08881 1/20 0.41
PIK3CA P42336 2/20 0.41
ROCK2 O75116 1/20 0.41
EGLN1 Q9GZT9 1/20 0.40
PTAFR P25105 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9247566 0.91 PTGER4 (0.49) NLRP3JAK2JAK1TYK2JAK3
SCHEMBL9251311 0.88 MEN1 (0.43) PTGER4MEN1KMT2ANAMPTPIK3CA
SCHEMBL9256202 0.83 JAK2 (0.55) JAK2JAK1TYK2JAK3PTGER4
SCHEMBL9247747 0.83 PTGER4 (0.49) JAK2JAK1TYK2JAK3PTGER4
SCHEMBL9251402 0.82 PTGER4 (0.51) JAK2JAK1TYK2JAK3PTGER4
SCHEMBL9255968 0.81 HDAC1 (0.51) JAK2JAK1TYK2JAK3PTGER4
SCHEMBL9253691 0.81 JAK2 (0.60) JAK2JAK1TYK2JAK3PTGER4
SCHEMBL9255820 0.81 ADORA2A (0.54) JAK2JAK1TYK2JAK3PTGER4
Hydrochloric Acid SCHEMBL9254291 0.81 JAK2 (0.59) JAK2JAK1TYK2JAK3PTGER4
SCHEMBL9256255 0.80 PTGER4 (0.50) JAK2JAK1TYK2JAK3PTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed