SCHEMBL9255752

SCHEMBL9255752

C=C[C@H]1CC[C@H]([C@H]2CC[C@H](CCc3ccc(Cl)c(F)c3)CC2)CC1

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PROKR1 Q8TCW9 3/20 0.34
FPR2 P25090 2/20 0.34
HTR2A P28223 3/20 0.32
HTR2C P28335 3/20 0.32
MAOB P27338 3/20 0.30
MAOA P21397 1/20 0.30
PNMT P11086 1/20 0.30
TAAR1 Q96RJ0 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30
KCNH2 Q12809 1/20 0.30
SIGMAR1 Q99720 3/20 0.30
DRD4 P21917 1/20 0.30
OPRL1 P41146 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9255736 1.00 PROKR1 (0.34) PROKR1FPR2HTR2AHTR2CMAOB
SCHEMBL9255744 1.00 PROKR1 (0.34) PROKR1FPR2HTR2AHTR2CMAOB
SCHEMBL9246826 0.90 PROKR1 (0.34) PROKR1FPR2HTR2AHTR2CMAOB
SCHEMBL9246820 0.90 PROKR1 (0.34) PROKR1FPR2HTR2AHTR2CMAOB
SCHEMBL9246812 0.90 PROKR1 (0.34) PROKR1FPR2HTR2AHTR2CMAOB
SCHEMBL9481182 0.88 SLC6A2 (0.35) MAOBMAOASLC6A2SLC6A4SLC6A3
SCHEMBL9481211 0.88 SLC6A2 (0.35) MAOBMAOASLC6A2SLC6A4SLC6A3
SCHEMBL9481205 0.88 SLC6A2 (0.35) MAOBMAOASLC6A2SLC6A4SLC6A3
SCHEMBL9262567 0.88 PNMT (0.39) PNMTTAAR1SIGMAR1
SCHEMBL9262557 0.88 PNMT (0.39) PNMTTAAR1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458176-B1 Bicyclohexyl derivatives HOFFMANN LA ROCHE (CH) 1995-08-02 EP disclosed
US-5174921-A BICYCLOHEXYL DERIVATIVES HOFFMANN-LA ROCHE INC. (US) 1992-12-29 US disclosed
EP-0458176-A1 Bicyclohexyl derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-11-27 EP disclosed