SCHEMBL9256419

SCHEMBL9256419

O=[N+]([O-])c1ccc2c(c1)CNC=C2

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PNMT P11086 8/20 0.47
ADRA2A P08913 6/20 0.47
PARP1 P09874 1/20 0.44
ADRA2B P18089 3/20 0.44
ADRA2C P18825 3/20 0.44
TDP2 O95551 1/20 0.42
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
STAT3 P40763 1/20 0.41
MTOR P42345 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
HIF1A Q16665 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7208524 0.74 PNMT (0.53) PNMTADRA2AADRA2BADRA2CTDP2
SCHEMBL17667571 0.74 MEN1 (0.58) PNMTADRA2AADRA2BADRA2CTDP2
SCHEMBL17667569 0.74 MEN1 (0.58) PNMTADRA2AADRA2BADRA2CTDP2
SCHEMBL7863751 0.74 CA9 (0.45) PNMTADRA2AADRA2BADRA2CTDP2
SCHEMBL1779718 0.71 PNMT (0.45) PNMTADRA2AADRA2BADRA2CTDP2
SCHEMBL16294213 0.70 PARP1 (0.44) PNMTADRA2APARP1ADRA2BADRA2C
SCHEMBL4976676 0.69 PARP1 (0.52) PARP1
SCHEMBL383577 0.69 PNMT (0.74) PNMTADRA2AADRA2BADRA2C
SCHEMBL7382123 0.69 PARP1 (0.52) PARP1
SCHEMBL11142660 0.69 PARP1 (0.52) PARP1MEN1NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107501099-A The adjusting control agent of ATP combination cassette transporters 沃泰克斯药物股份有限公司 2017-12-22 CN disclosed
CN-104788328-B The adjusting control agent of ATP combination cassette transporters 沃泰克斯药物股份有限公司 2017-09-12 CN disclosed
CN-103641765-B ATP-combines the adjusting control agent of cassette transporters 沃泰克斯药物股份有限公司 2016-08-17 CN disclosed
CN-101935301-A Modulators of ATP-binding cassette transporters VERTEX PHARMA 2011-01-05 CN disclosed
CN-101891680-A The adjusting control agent of ATP- combination cassette transporters VERTEX PHARMA 2010-11-24 CN disclosed
US-5464871-A Aromatic amides OCTAMER, INC. (US) 1995-11-07 US disclosed