SCHEMBL9259538

SCHEMBL9259538

O=[C]N(c1ccccc1)c1cccnc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 5/20 0.50
KCNN4 O15554 3/20 0.43
HTT P42858 1/20 0.41
GAA P10253 2/20 0.40
TSHR P16473 1/20 0.40
ALDH1A1 P00352 2/20 0.38
APP P05067 1/20 0.38
HCAR3 P49019 1/20 0.38
HCAR2 Q8TDS4 1/20 0.38
CFTR P13569 1/20 0.38
SLC6A2 P23975 1/20 0.38
SLC6A4 P31645 1/20 0.38
SLC6A3 Q01959 1/20 0.38
GOPC Q9HD26 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
CYP19A1 P11511 1/20 0.38
NPC1 O15118 1/20 0.37
PKM P14618 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9276044 0.82 KMT2A (0.43) KCNA5HTTALDH1A1SLC6A2SLC6A4
SCHEMBL104821 0.81 ALDH1A1 (0.42) HTTGAATSHRALDH1A1NPC1
SCHEMBL348708 0.74 KCNA5 (0.43) KCNA5KCNN4HTTGAAALDH1A1
SCHEMBL6225489 0.74 USP2 (0.35) KCNA5KCNN4HTTALDH1A1CYP1A2
SCHEMBL6328963 0.73 KCNA5 (0.53) KCNA5KCNN4HTTGAATSHR
SCHEMBL16484704 0.73 KCNA5 (0.53) KCNA5KCNN4HTTGAATSHR
SCHEMBL9183264 0.71 ALDH1A1 (0.44) KCNA5KCNN4HTTTSHRALDH1A1
SCHEMBL5511544 0.70 HTT (0.45) KCNA5KCNN4HTTALDH1A1CYP2A6
SCHEMBL5075470 0.69 KCNA5 (0.50) KCNA5KCNN4HTTGAAALDH1A1
SCHEMBL4234956 0.69 KCNA5 (0.50) KCNA5KCNN4HTTGAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5405843-A Anticancer drug potentiators MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1995-04-11 US disclosed
EP-0363212-B1 Novel heterocyclic compounds and anticancer-drug reinforcing agents containing them as effective components MITSUI TOATSU CHEMICALS (JP) 1995-01-04 EP disclosed
US-5204348-A Quinoline derivatives MITSUI TOATSU CHEMICALS INC. (JP) 1993-04-20 US disclosed
US-5112817-A Anticancer Drug Potentiators MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1992-05-12 US disclosed
EP-0363212-A2 Novel heterocyclic compounds and anticancer-drug reinforcing agents containing them as effective components MITSUI TOATSU CHEMICALS, Inc. (JP) 1990-04-11 EP disclosed