SCHEMBL9259986

SCHEMBL9259986

C=CC(N)C(=O)c1ccc(O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH5A1 P51649 1/20 0.50
ABAT P80404 1/20 0.50
PDPK1 O15530 1/20 0.46
MAPT P10636 3/20 0.43
LMNA P02545 2/20 0.43
HTT P42858 2/20 0.43
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43
PKM P14618 1/20 0.43
HPGD P15428 1/20 0.43
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CA12 O43570 2/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
CA14 Q9ULX7 2/20 0.41
CA3 P07451 1/20 0.41
TYR P14679 1/20 0.41
DRD1 P21728 1/20 0.41
CA4 P22748 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL45332 0.82 AKT1 (0.48) MAPTLMNACA1CA2CA12
Hydroxylated Completely Delakylated Diethylpropion SCHEMBL27460979 0.72 CA1 (0.50) PDPK1MAPTLMNAHTTESR1
Hydroxylated Completely Delakylated Diethylpropion SCHEMBL5319402 0.72 CA1 (0.50) PDPK1MAPTLMNAHTTESR1
SCHEMBL1223467 0.71 CA1 (0.50) PDPK1MAPTLMNAHTTESR1
Hydroxylated Completely Delakylated Diethylpropion SCHEMBL5172799 0.71 CA1 (0.48) PDPK1MAPTLMNAHTTESR1
SCHEMBL9658758 0.69 CA1 (0.47) PDPK1MAPTLMNAHTTESR1
SCHEMBL11538990 0.68 PDPK1 (0.50) ALDH5A1ABATPDPK1MAPTLMNA
SCHEMBL6654144 0.68 PDPK1 (0.46) PDPK1MAPTLMNAHTTESR1
SCHEMBL6654142 0.68 PDPK1 (0.46) PDPK1MAPTLMNAHTTESR1
SCHEMBL2574988 0.68 PDPK1 (0.46) PDPK1MAPTLMNAHTTESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431871-B1 A process for the preparation of ketones FINE ORGANICS LTD (GB) 1995-06-07 EP claimed
US-5276191-A Reacting phenol with a nitrile in presence of Lewis acid catalyst in nitroalkane solvent to produce aminoalkyl para-hydroxyphenyl ketone FINE ORGANICS LIMITED (GB) 1994-01-04 US claimed
EP-0431871-A2 A process for the preparation of ketones FINE ORGANICS LIMITED (GB) 1991-06-12 EP claimed
JP-3279351-A None JP disclosed
EP-0431871-B1 A process for the preparation of ketones FINE ORGANICS LTD (GB) 1995-06-07 EP disclosed
US-5276191-A Reacting phenol with a nitrile in presence of Lewis acid catalyst in nitroalkane solvent to produce aminoalkyl para-hydroxyphenyl ketone FINE ORGANICS LIMITED (GB) 1994-01-04 US disclosed
US-5276191-A Reacting phenol with a nitrile in presence of Lewis acid catalyst in nitroalkane solvent to produce aminoalkyl para-hydroxyphenyl ketone FINE ORGANICS LIMITED (GB) 1994-01-04 US disclosed
JP-H03279351-A PREPARATION OF KETONE FINE ORGANICS LTD 1991-12-10 JP disclosed
EP-0431871-A2 A process for the preparation of ketones FINE ORGANICS LIMITED (GB) 1991-06-12 EP disclosed
EP-0431871-A2 A process for the preparation of ketones FINE ORGANICS LIMITED (GB) 1991-06-12 EP disclosed