SCHEMBL9263181

SCHEMBL9263181

Fc1ccc2nc[nH]c(=S)c2c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.64
IP6K1 Q92551 2/20 0.45
IP6K3 Q96PC2 1/20 0.45
QPCT Q16769 1/20 0.41
PDPK1 O15530 1/20 0.39
CHEK1 O14757 2/20 0.39
PIM1 P11309 1/20 0.39
AKT1 P31749 1/20 0.39
FLT3 P36888 1/20 0.39
PIM3 Q86V86 1/20 0.39
PPARG P37231 1/20 0.38
RAB9A P51151 1/20 0.38
NCOA2 Q15596 1/20 0.38
NCOA1 Q15788 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
TYMS P04818 2/20 0.36
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
USP10 Q14694 1/20 0.36
PIK3C3 Q8NEB9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27828038 0.78 PIM1 (0.64) PARP1QPCTCHEK1PIM1AKT1
SCHEMBL29709603 0.78 PARP1 (1.00) PARP1IP6K1IP6K3PDPK1CHEK1
SCHEMBL2191067 0.78 PARP1 (1.00) PARP1IP6K1IP6K3PDPK1CHEK1
Hydrochloric Acid SCHEMBL30141968 0.76 PARP1 (0.96) PARP1IP6K1IP6K3PDPK1CHEK1
SCHEMBL914338 0.72 PDPK1 (0.59) PARP1IP6K1IP6K3PDPK1PPARG
SCHEMBL903277 0.72 PRKCI (0.59) PARP1QPCTPOLBHTTSMN1; SMN2
SCHEMBL21025330 0.70 IP6K1 (0.40) PARP1IP6K1IP6K3QPCTCHEK1
SCHEMBL13948932 0.69 MAPT (0.48) QPCTPPARGRAB9ANCOA2NCOA1
SCHEMBL903276 0.68 PARP1 (0.52) PARP1IP6K1IP6K3QPCTPDPK1
SCHEMBL6836398 0.68 KDM4A (0.49) PARP1IP6K1QPCTPDPK1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5387585-A Treating epilepsy, anxiety, sleep disorders, schizophrnia, senile dementia HOFFMANN-LA ROCHE INC. (US) 1995-02-07 US disclosed